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3-[2-(4-benzylpiperidin-1-yl)-2-oxoethyl]-4-(2-phenylethyl)piperazin-2-one
N-({1-[2-(pyridin-2-yl)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
[2-(2-{3,9-diazaspiro[5.5]undecan-3-ylmethyl}phenoxy)ethyl]dimethylamine
N-[(4-chlorophenyl)(phenyl)methyl]-5-oxopyrrolidine-3-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-{2-[(2,4-dimethylphenyl)carbamoyl]ethyl}-2-[(3-methoxyphenyl)amino]butanamide
1-(2-aminoethyl)-N-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
9-(2H-1,3-benzodioxol-5-yl)-15-methyl-12-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4-(trifluoromethyl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-({[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}amino)ethan-1-one
methyl 6-[(4-formyl-1,4-diazepan-1-yl)methyl]-3-[(2E)-3-phenylprop-2-enamido]thieno[2,3-b]pyridine-2-carboxylate
3-[(3R,4S)-1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-(3-methoxyphenyl)piperidin-4-amine
5-({[2-(azepan-1-yl)ethyl](ethyl)amino}methyl)-N-ethylpyrimidin-2-amine
N'-(2,4-dimethylphenyl)-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]propanediamide
ethyl 1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxylate
(2S)-2-amino-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-phenylethan-1-one
2-{1-[(5-methylfuran-2-yl)methyl]-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
2-{1-[(2-ethoxyphenyl)methyl]-4-[(3-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
3-(methylsulfanyl)-N-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
(3R,4S)-4-[ethyl({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})amino]oxolan-3-ol
N-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-N-methyloxan-4-amine
N-cyclopentyl-2,3,4-trimethoxy-N-{[4-(oxolan-3-yloxy)phenyl]methyl}benzamide
6-methyl-3-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
(2S)-N-[(1R)-1-(2-fluorophenyl)ethyl]-1-(piperidin-4-yl)pyrrolidine-2-carboxamide
2-{[(1R,5R)-3-(dimethylsulfamoyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzoic acid
(1R,5S)-N-[4-(pyridin-3-yloxy)phenyl]-6-azabicyclo[3.2.1]octane-6-carboxamide
N-[(3S,4R)-1-(3-aminothiophene-2-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
N-[(5-methylpyrazin-2-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-2-(1,4-dimethylpiperazin-2-yl)acetamide
4-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}-1-(3-fluorobenzoyl)piperidine
2-(1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine-3-carbonyl)pyridine
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(dimethylamino)ethyl]-N-ethylacetamide
methyl 4-({4-[5-(2-methoxybenzamido)-1H-pyrazol-1-yl]piperidin-1-yl}methyl)benzoate
4-(methylsulfanyl)-2-[(3-propanamidophenyl)formamido]butanoic acid
N-{1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-4-yl}methanesulfonamide
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
N5-[2-methoxy-2-(thiophen-2-yl)ethyl]-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-{3-[1-(4-fluoro-3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propyl}-1H-pyrazole
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
6-chloro-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-1-methyl-1H-indole-2-carboxamide
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)-4-{[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]amino}pyrrolidine-2-carboxamide
2,5-dimethoxy-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzamide
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidine
2-[1-(cyclohexylmethyl)-4-[2-(4-fluorophenoxy)ethyl]piperazin-2-yl]ethan-1-ol
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropylpyrazolo[1,5-a]pyrimidine-2-carboxamide
N-cyclopropyl-3-(2-methoxyphenyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
2-{imidazo[1,2-a]pyridin-3-yl}-N-[(2-phenoxypyridin-3-yl)methyl]acetamide
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-propylacetamide
1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-amine