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(2S,4S)-1-cyclopentyl-4-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamido]-N-ethylpyrrolidine-2-carboxamide
3-{1-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}quinoline
1-(4-benzylpiperazin-1-yl)-3-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-3-yl}propan-1-one
2-methyl-5-{4-[4-(3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-1-yl)benzoyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
2-{3-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
5-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-5-oxopentanamide
N-cycloheptyl-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
3-(4-methoxyphenyl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]acetamide
2-acetamido-N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
6-ethyl-2-methyl-N-[3-(4H-1,2,4-triazol-4-yl)propyl]quinoline-4-carboxamide
2-methyl-4-{3-[2-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenyl}pyrimidine
(4-{[5-(1-ethyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}phenyl)methanol
N-cyclopropyl-1-[(1s,4s)-4-[(1,3-benzothiazol-2-ylmethyl)amino]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-(1-{1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
1-(3-methoxyphenyl)-6-methyl-4-[(3-methylthiophen-2-yl)methyl]piperazin-2-one
1-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
1-({5-[1-(4-fluorophenyl)-2,2-dimethylcyclopropyl]-1,2,4-oxadiazol-3-yl}methyl)-4-methylpiperazine
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
2-methyl-2-phenyl-N-[4-(1H-pyrazol-1-yl)butan-2-yl]propanamide
4-({1-[(5-hydroxy-2-methoxyphenyl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
2-(1H-indol-3-yl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
2-(2-methylfuran-3-carbonyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidin-1-yl]-2-[2-(trifluoromethyl)phenyl]ethan-1-one
4-butyl-11-({[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-[3-(2-methylpropyl)-1,2-oxazole-5-amido]pyrrolidine-3-carboxylic acid
methyl (2S,4R)-1-[(4-ethylphenyl)methyl]-4-{2-[4-(trifluoromethyl)phenyl]benzamido}pyrrolidine-2-carboxylate
6-fluoro-2-[({[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}amino)methyl]quinolin-4-ol
2-[5-chloro-2-(propan-2-yloxy)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3R)-3,4,4-trimethyl-1-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]pyrrolidin-3-ol
N-(1-hydroxybutan-2-yl)-2-methyl-N-(pyridin-3-ylmethyl)furan-3-carboxamide
N-(1-{7-[(4-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
2-{4-[2-(2-phenylethyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
N-(3-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}propyl)-N,3-dimethyl-1,2-oxazole-5-carboxamide
7-chloro-3-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]quinolin-4-ol
5-chloro-3-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
3-(3-chlorophenyl)-6-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
5-methyl-1-propyl-N-[1-(1,3-thiazol-5-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
N-benzyl-2-[2,5-dioxo-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-(2-hydroxyethyl)acetamide
1-(4-benzylpiperidin-1-yl)-3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]propan-1-one
1-(4-ethylphenyl)-3-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}urea
(1R,2S)-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-2-propyl-N-(pyridin-4-ylmethyl)cyclopropane-1-carboxamide
2-methyl-5-(4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
1-[2-(dimethylamino)-6-(1H-1,2,3-triazole-5-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
(1S,5R)-6-(propane-1-sulfonyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
3-[2-(3,4-difluorophenyl)ethyl]-1-(1H-pyrrole-2-carbonyl)piperidine
N-({1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-2-(2-oxo-1,2-dihydroquinoxalin-1-yl)acetamide
5-(2-methyl-1-benzofuran-5-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
7-(oxan-4-yl)-2-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one