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3-{[(1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-yl)oxy]methyl}pyridine
8-[(1-benzyl-1H-imidazol-5-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
1-[(2-fluorophenyl)methyl]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
9-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[(2,4-difluorophenyl)methyl]-1-(4-methylpyrimidin-2-yl)piperidine-3-carboxylic acid
methyl 3-({1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)propanoate
N-[2-(dimethylsulfamoyl)ethyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(3-hydroxyquinoxalin-2-yl)propanamide
1-(1-methanesulfonylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
(3S,4S)-4-(morpholin-4-yl)-1-(pyridin-4-ylmethyl)pyrrolidin-3-ol
N-(furan-2-ylmethyl)-2-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]acetamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-[(dimethyl-1,3-thiazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
2-(5-fluoro-2-methoxyphenyl)-2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}acetic acid
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}bis(prop-2-en-1-yl)amine
(3R,4S)-3,4-dimethyl-1-[1-methyl-5-(trifluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-4-ol
8-[(2,3-difluoro-4-methylphenyl)methyl]-8-azaspiro[4.5]decane-7,9-dione
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
3-(3-acetylphenyl)-6-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-(3-methylbut-2-en-1-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-butyl-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]acetamide
N,1-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
6-[3-(ethylsulfanyl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-(1-methyl-1H-pyrazol-4-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}propanamide
N-[1-(methylcarbamoyl)cyclohexyl]-3-(piperidin-3-yl)benzamide
2-({7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)phenol
[(3S,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]methanol
1-(2-ethylpyrimidine-5-carbonyl)azocane
2-(3-methyl-1H-pyrazole-4-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
ethyl 1-benzyl-5-[3-(thiophen-2-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
3-cyclopropyl-5-{pyrazolo[1,5-a]pyridin-3-yl}-1H-1,2,4-triazole
1,3-dimethyl-2,6-dioxo-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-{[(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}benzonitrile
N3-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-methyl-N-{[8-(naphthalen-2-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}propanamide
2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
5-butyl-N-ethyl-N-[(3R,4R)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]pyridine-2-carboxamide
2-[2-(benzyloxy)phenyl]-6-methylpyridine-3-carboxamide
1-methyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(2S,4S)-1-methyl-4-(2,3,6-trimethylquinoline-4-amido)pyrrolidine-2-carboxylic acid
1-{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]azetidin-3-yl}-3,5-dimethyl-1H-pyrazole
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-5-(trifluoromethyl)pyridine
N-ethyl-N-methyl-5-{1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(pyrrolidin-1-yl)piperidine
2-(dimethylamino)-2-(2-fluorophenyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
5-methoxy-2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-4H-pyran-4-one
5-(6-methoxypyrimidin-4-yl)-2-methylquinoline
(1S,5R)-6-(cyclopropylmethyl)-3-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane