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3-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}pyridine
1-(4-fluorophenyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,4-diazepane
2-{2-[(2-methylphenyl)sulfanyl]acetyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl 2-{N-methyl-1-[2-(phenoxymethyl)-1,3-oxazol-4-yl]formamido}acetate
5-ethyl-1'-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]propan-1-one
5-ethyl-1'-(4-phenyl-1,3-thiazol-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
{[2,5-dimethyl-1-(4-methylpyridin-2-yl)-1H-pyrrol-3-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
2-(4-benzyl-3-ethyl-5-oxo-1,4-diazepane-1-carbonyl)benzonitrile
3-cyclohexyl-1-(1,4-oxazepan-6-ylmethyl)urea
methyl 1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carboxylate
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(3-phenylpropyl)-1,4-diazepane
({1-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)(methyl)propylamine
2-ethyl-8-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
3-{3-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-3-oxopropyl}-3,4-dihydroquinazolin-4-one
2-(pyridin-4-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2,4-dimethylpyrimidine-5-carboxamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1-methylpiperidine-4-carboxamide
6-methyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-5-carboxamide
1-[2-(1-methyl-1H-pyrazol-3-yl)piperidin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
{1-[1-(3-fluorobenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}(methyl)(pyridin-2-ylmethyl)amine
2-({[(1R,3R)-3-aminocyclopentyl]amino}methyl)-6-methylquinolin-4-ol
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
{[4-(1H-imidazol-1-yl)phenyl]methyl}(methyl)[(3-methylpyridin-4-yl)methyl]amine
1-[(4aR,8aS)-6-[4-(trifluoromethyl)benzoyl]-decahydro-1,6-naphthyridin-1-yl]butan-1-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(2S)-pyrrolidin-2-ylmethyl]-1,3-oxazole-4-carboxamide
4-[(1-cycloheptylpiperidin-4-yl)oxy]-N-(pyridin-4-ylmethyl)benzamide
N-[(2-ethoxy-3-methoxyphenyl)methyl]-N-methyl-2-[methyl(piperidin-4-yl)amino]acetamide
3-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
N-[1-(cyclohex-1-en-1-yl)ethyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-phenoxybutan-1-one
1-({2-[2-hydroxy-3-(pyrrolidin-1-yl)propoxy]-4-methoxyphenyl}methyl)-4-(hydroxymethyl)piperidin-4-ol
2,4-dimethyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}pyrimidine-5-carboxamide
7-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
2-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)acetamide
N-[(1S,2R)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-yl]-2-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
6-methyl-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]imidazo[1,2-a]pyridine-2-carboxamide
1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
4-fluoro-N-({1-[2-(pyridin-2-ylsulfanyl)acetyl]piperidin-3-yl}methyl)benzamide
2-(2-phenyl-1H-imidazol-1-yl)-1-[(2S)-2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]ethan-1-one
2-[(3,5-difluorophenyl)methyl]-8-(pyrimidin-5-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
(2R,3S,6R)-5-[(1R,5S,6R)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-[(2-chlorophenyl)methyl]-3-(2-methoxyethyl)-5-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
(3R)-N-(2-methoxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(1H-pyrrole-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
ethyl 3-[(2-fluorophenyl)methyl]-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidine-3-carboxylate