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N-(cyclohex-1-en-1-ylmethyl)-2-{4-[2-(2-oxopiperidin-1-yl)acetyl]morpholin-3-yl}acetamide
3-acetyl-N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-1H-pyrazole-5-carboxamide
5-[benzyl(methyl)amino]-2-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
ethyl 2-(1-{3-[(4-fluorophenyl)formamido]propanoyl}piperidin-2-yl)acetate
2-[(6-methoxypyridin-3-yl)methyl]-9-oxa-2-azaspiro[5.5]undecane
1-{1-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]propan-2-yl}-1H-1,3-benzodiazole
5-(azocane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-4-(2-fluoro-5-methylphenoxy)piperidine-4-carboxylic acid
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-methylacetamide
2-{4-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]piperazin-1-yl}-N-ethylacetamide
(4aS,8aR)-1-(2-aminoethyl)-6-{2-[(dimethylamino)methyl]benzoyl}-decahydro-1,6-naphthyridin-2-one
4-{1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]piperidin-3-yl}benzoic acid
1-{3-[3-(4-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxymethyl)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
2-chloro-4-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}phenol
(4aS,8aR)-1-(3-hydroxypropyl)-6-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
methyl 3-[2-(cyclohex-1-en-1-yl)acetyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(piperidin-1-yl)-3-[2-({[3-(pyridin-3-yloxy)propyl]amino}methyl)phenoxy]propan-2-ol
methyl(quinolin-6-ylmethyl){[4-({1-[3-(trifluoromethyl)benzenesulfonyl]piperidin-4-yl}oxy)phenyl]methyl}amine
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-2-methylpropanamide
1-[(3S)-3-ethylmorpholin-4-yl]-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
5-methyl-1-(2-methylphenyl)-4-[2-(methylsulfanyl)benzoyl]piperazin-2-one
4-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-1-(4-methylphenyl)piperazin-2-one
7-(2,6-dimethoxypyridine-3-carbonyl)-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(3-cyclopentylpropanoyl)-9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-(3-{[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]methyl}phenyl)-5-(pyrrolidin-1-yl)pyridazine
N-cyclopentyl-3-fluoro-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}benzene-1-sulfonamide
[4-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)oxan-4-yl]methanol
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)acetamide
N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
2-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-6-methoxy-1,2,3,4-tetrahydroisoquinoline
5-fluoro-1-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-indole-2-carboxamide
N-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-5-ethyl-2-methylpyrimidin-4-amine
5-(2-fluorophenyl)-2-(pyridin-3-yl)-4-[1-(thiophene-3-carbonyl)piperidin-3-yl]pyrimidine
3-ethoxy-N-[1-(4-fluorophenyl)-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]propanamide
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(methylsulfanyl)ethan-1-one
2-[4-(2-phenylpyrrolidine-1-carbonyl)piperidin-1-yl]acetamide
8-chloro-2-(furan-2-yl)-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-methylquinoline-4-carboxamide
ethyl 2-(4-{[(2S)-4-methyl-2-phenylpiperazine-1-carbonyl]amino}phenyl)acetate
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-{[1-(phenoxymethyl)cyclopropyl]methyl}propanamide
N-[(2R,3R)-1'-(2-ethylbutyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(2S)-2-{imidazo[2,1-b][1,3]thiazol-6-ylformamido}-4-methanesulfonylbutanoic acid
6-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
(3S,4R)-4-(2-methoxyphenyl)-1-[3-(4-methylpiperazin-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
5-(propan-2-yl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-(3,3-diphenylpiperidine-1-carbonyl)-6-(methoxymethyl)pyridine
N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
N-{3-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]phenyl}acetamide
4-(3-{1-[(1-methyl-1H-imidazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)isoquinoline