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3-({ethyl[(5-methylfuran-2-yl)methyl]amino}methyl)-7-methyl-1,2-dihydroquinolin-2-one
3-[methyl(1,3-thiazol-2-ylmethyl)sulfamoyl]-N-(pyridin-3-yl)benzamide
3-methyl-N-[(3R,5S)-1-methyl-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-4-oxo-3,4-dihydroquinazoline-7-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-6-[3-(1H-pyrazol-1-yl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
2-methyl-9-({2-oxo-3-oxatricyclo[7.3.1.05,13]trideca-1(12),5(13),6,8,10-pentaen-8-yl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-N-(2-methylpropyl)-3-[2-(pyridin-2-yl)-1H-imidazol-1-yl]benzamide
4-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]-2,3,6-trimethylquinoline
3-{[2-(butan-2-yl)-1H-imidazol-1-yl]methyl}-5-ethyl-1,2,4-oxadiazole
N-{[4-(dimethylsulfamoyl)phenyl]methyl}-2-(2,5-dioxoimidazolidin-1-yl)acetamide
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methylpyridin-2-yl)methyl]acetamide
dimethyl({4-[1-(3-methylbenzoyl)piperidin-2-yl]phenyl}methyl)amine
1-ethyl-N-(2-methylpropyl)-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-3-(3-methylpiperidin-1-yl)propanamide
(2R)-2-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyrrolidine
2-[1-(3-methylbut-2-en-1-yl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
2-(2,4-dimethoxyphenyl)-8-methoxy-5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
7-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(3S,4R)-1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
N-(1-carbamoylcyclohexyl)-3,5,7-trimethyl-1H-indole-2-carboxamide
2-{[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]methyl}-5,8-dimethyl-1,4-dihydroquinolin-4-one
ethyl 4-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)piperazine-1-carboxylate
(1R,5R)-6-[(3-chloro-4-fluorophenyl)methyl]-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane
5-[2-(propan-2-yl)-1,3-benzoxazol-5-yl]quinoline
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
7-(cyclobutylmethyl)-2-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-2,7-diazaspiro[4.5]decan-6-one
8-{[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}quinoline
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]acetamide
5-acetyl-N-(2-propoxyethyl)thiophene-3-carboxamide
3,5-dimethyl-N,N-bis(prop-2-en-1-yl)-1-benzofuran-2-carboxamide
2-amino-4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
N,3,4-trimethyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5-sulfamoylbenzamide
3-{1-[(2-chlorophenyl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
1-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]-2-(4-methanesulfonylphenyl)ethan-1-one
2-(1-methylpyrrolidin-3-yl)-9-(5-methylthiophene-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonyl}azepane
N,2-dimethyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-6-(piperidin-3-yl)pyrimidin-4-amine
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-5-phenylpentanamide
3-(3-methyl-1H-pyrazol-1-yl)-N-{[7-(pyridin-3-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}propanamide
1-[2-(methylsulfanyl)ethyl]-4-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperazine
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-4-(2-methylphenyl)-1,4-diazepane
N-[(2-chloro-6-fluorophenyl)methyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
ethyl 4-[(3-fluorophenyl)methyl]-1-[1-(pyridin-3-yl)propan-2-yl]piperidine-4-carboxylate
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[4-(methylsulfanyl)phenyl]methyl}amine
N-ethyl-3-methyl-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]aniline
N-[(2-chlorophenyl)methyl]-3-[1-(3-acetamidobenzoyl)piperidin-3-yl]propanamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-methyl-N-(naphthalen-1-ylmethyl)acetamide
5-(5-{[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)-3-methyl-1,2-oxazole
2-(4-fluorophenyl)-1-[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]azetidine
4,6-dimethyl-2-[({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)amino]pyridine-3-carbonitrile