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2-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-2-(thiophen-3-yl)acetamide
3-{[1-methyl-6-oxo-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
[(6-fluoroquinolin-2-yl)methyl](methyl)[4-(morpholin-4-yl)butyl]amine
2-({3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
2-(dimethyl-1,2-oxazol-4-yl)-N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)acetamide
5-methyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]pyrimidin-2-amine
1-{2-[4-(2-amino-6-methylpyrimidin-4-yl)piperazin-1-yl]pyrimidin-4-yl}pyrrolidin-3-ol
2-amino-6-(3,4-dichlorophenyl)-4-(oxolan-3-yl)pyridine-3-carbonitrile
N-(2H-1,3-benzodioxol-5-yl)-3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}benzamide
3-{2-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}imidazolidine-2,4-dione
6-(4-methyl-3-oxopiperazin-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-{2-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]ethyl}-2-methylpropanamide
N-(2-hydroxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(morpholin-4-yl)benzamide
N-[(3S,4R)-1-{2-[(dimethylcarbamoyl)amino]acetyl}-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-N-{[2-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-methyl-7-{[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-2H-chromen-2-one
4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-2-(pyridin-3-yl)morpholine
1-(2,3-dihydro-1-benzothiophene-2-carbonyl)-4-(furan-3-carbonyl)-1,4-diazepane
1-{2-[5-(2,4-dimethoxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyrrolidin-2-one
[(5-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}furan-2-yl)methyl]dimethylamine
3-[(dimethylamino)methyl]-1-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]pyrrolidin-3-ol
(3aR,6aR)-2-[2-(methylsulfanyl)acetyl]-5-(pyridin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-benzyl-3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]-3-(2-methylphenyl)pyrrolidine-2,5-dione
1'-(6-aminopyridine-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-benzyl-8-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-{[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]amino}-N,N-dimethylpyrazine-2-carboxamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}piperidin-2-one
9-[(1S,3R)-3-aminocyclopentanecarbonyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
5-fluoro-1,3-dimethyl-N-(2-methylpropyl)-N-(pyridin-4-ylmethyl)-1H-indole-2-carboxamide
4-[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]-N,N-dimethylbutanamide
2-[(2-methoxyethyl)(methyl)amino]-2-[4-(propan-2-yl)phenyl]acetic acid
N-(3,4-difluorophenyl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-3-amine
1-methyl-2-oxo-8-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
[1-(2,6-dimethylquinoline-4-carbonyl)azepan-2-yl]methanol
N-(2-phenoxyphenyl)-2-(trifluoromethyl)morpholine-4-carboxamide
(2S,4R)-1-[(2,6-difluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-(2-methyl-1,3-benzothiazol-5-yl)pyrrolidine-2-carboxamide
N-(1-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
(3aS,6aR)-5-(5-chloropyridin-2-yl)-3-[3-(4-methoxyphenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(4-methoxyphenyl)propanamide
1-methyl-3-[2-oxo-2-(piperidin-1-yl)ethyl]-1H,2H,3H-imidazo[4,5-c]pyridin-2-one
5-(4-fluoro-2-methylphenyl)-1-(oxolan-2-ylmethyl)-4-phenyl-1H-imidazole
methyl 4-{[(4-methyl-5-{1-[3-(6-methylpyridin-2-yl)propyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-yl)amino]methyl}benzoate
2-methoxy-1-{4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}ethan-1-one
3-(3-chloro-1,2-oxazol-5-yl)-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
2,8-dimethyl-N-[3-(4H-1,2,4-triazol-4-yl)propyl]quinoline-4-carboxamide
2-{[(5-hydroxypentyl)amino]methyl}-6,8-dimethylquinolin-4-ol
(3aR,6aR)-2-(cyclopentylcarbamoyl)-5-(pyridin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[2-(dimethylamino)ethyl]-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide