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4-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-4-oxobutane-1-sulfonamide
1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]pyrrolidin-3-yl]methanol
2-(2-methoxyethyl)-8-(2-methyl-1-benzofuran-7-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[4-(aminomethyl)phenyl]methyl}-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[1-(3-methylbutyl)-1H-1,3-benzodiazol-2-yl]methyl})amine
2-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-1H-indole
2-(4-methylpentyl)-4-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]morpholine
methyl[(3-methylpyridin-4-yl)methyl][(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
2-chloro-N-({1-[2-(methylsulfanyl)benzoyl]piperidin-3-yl}methyl)benzamide
4-{[5-(methoxymethyl)furan-2-yl]methyl}-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](ethyl)[(4-methyl-1H-imidazol-5-yl)methyl]amine
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(5-methyl-1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decane
2-amino-6-(2,6-difluorophenyl)-4-(2-methoxypyrimidin-5-yl)pyridine-3-carbonitrile
(1R,2R,6S,7S)-4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-10-oxa-4-azatricyclo[5.2.1.02,6]decane
1-[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]-3-(2-methyl-1-benzofuran-5-yl)urea
N-(1-{1-[(4-fluoro-2-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
(3aR,6aR)-2-(3-chloro-2-methylbenzoyl)-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-amino-6-(1-methyl-1H-pyrrol-3-yl)-4-[2-(prop-2-en-1-yloxy)phenyl]pyridine-3-carbonitrile
4-{[1-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}-N-ethylpiperidine-1-carboxamide
6-hydroxy-N-{1-oxaspiro[4.4]nonan-3-yl}pyridine-2-carboxamide
(3R,4S)-4-({[3-(cyclopentyloxy)phenyl]methyl}(methyl)amino)oxolan-3-ol
1-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-4-methylpiperazine
7-(2-methoxyethyl)-2-[6-(trifluoromethyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclobutanecarboxamide
2-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindole-2-carbonyl]-1,4-dihydroquinolin-4-one
1-{4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}isoquinoline
2-[2-(1H-imidazol-1-yl)ethyl]-1-[(3-methylthiophen-2-yl)methyl]piperidine
6-[(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
7-[6-(piperidine-1-carbonyl)pyrazin-2-yl]-2,7-diazaspiro[4.4]nonane-1,3-dione
5-amino-3-[1-(pyridin-4-yl)-1H-pyrrol-2-yl]-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
2-{1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,3-triazol-4-yl}quinoline
6-{3,9-diazaspiro[5.6]dodecane-9-carbonyl}-1,2,3,4-tetrahydroquinoxaline-2,3-dione
ethyl 4-[7-(1-hydroxy-3-phenylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidine-1-carboxylate
1-(2-methoxyphenyl)-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
2-{2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamido}-N-methylacetamide
5-methoxy-2-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
2-amino-3-ethyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(1-methylpyrrolidin-3-yl)-3-oxo-N-propyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
[3-(2-phenylethyl)-1-(9H-purin-6-yl)piperidin-3-yl]methanol
2-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-4H-chromen-4-one
1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(methylamino)ethan-1-one
(1R)-1-[(4-methoxyphenyl)methyl]-2-(1-methyl-1H-pyrazole-5-carbonyl)-1,2,3,4,5,6,7,8-octahydroisoquinoline
1-(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperidin-4-ol
2-[1-(2-methylphenyl)-5-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)phenyl]-1H-1,2,4-triazol-3-yl]acetamide
2-({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-2-(4-fluorophenyl)ethan-1-ol
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(methylsulfanyl)propyl]acetamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-3-(2-oxoazepan-1-yl)propanamide
6-{3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]propanoyl}-2-methyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(4-methylphenyl)quinoline-4-carboxamide