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2,2,2-trifluoro-N-{2-[(2-oxo-2H-chromen-3-yl)formamido]ethyl}acetamide
6-ethyl-3-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-1,5-dimethyl-1,2-dihydropyridin-2-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[(3,4,5-trifluorophenyl)methyl]cyclopropanamine
(2E)-N-[(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)methyl]-3-phenylprop-2-enamide
7-(2,2-dimethylpropyl)-2-[(1-methyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(2-methoxyethoxy)ethan-1-one
methyl 3-[2-(4-fluorophenyl)acetamido]-6-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
N3-[3-(5-chloro-1H-1,3-benzodiazol-2-yl)propyl]piperidine-1,3-dicarboxamide
1-(3-methoxyphenyl)-4-(1-propylpiperidin-4-yl)piperazine
1-[(4-methoxyphenyl)methyl]-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
1-(pyrrolidine-1-sulfonyl)-2-[2-(thiophen-2-yl)ethyl]piperidine
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-(4-methoxyphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(quinolin-5-yl)pyridine-3-carboxamide
9-methoxy-4-[(4-methoxy-2,3-dimethylphenyl)methyl]-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(furan-3-ylmethyl)-3-(1,2-oxazinan-2-yl)propanamide
4-(2-methyl-1H-imidazol-1-yl)-1-[4-(piperidine-1-carbonyl)piperidin-1-yl]butan-1-one
3-(azepane-1-carbonyl)-5-(4-methylpiperidin-1-yl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyacetyl)pyrrolidin-3-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-[(4-phenyloxan-4-yl)methyl]acetamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
1-{5-[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
8-(2-hydroxypyridine-3-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[2-(dimethylamino)ethyl]-4-ethyl-3-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-cyclohexylethyl)-N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N,4-dimethyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-(4-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-2,5-dimethylpyrazine
(3R,4S)-1-[(4-methoxypiperidin-1-yl)sulfonyl]-4-phenylpyrrolidin-3-amine
N,N-diethyl-2-{4-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}acetamide
(3S)-1-{2-[(3-chlorophenyl)methyl]-1,3-benzoxazole-6-carbonyl}pyrrolidin-3-ol
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]propanamide
3-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1-methylpiperidine
(1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidin-3-yl)methanamine
2-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}-N,N-dimethylaniline
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
(2S,4S)-1-benzyl-N-methyl-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-[(1R,2S)-2-phenylcyclopropyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
N,N-dimethyl-3-[2-(morpholin-4-ylmethyl)phenyl]pyrazin-2-amine
1-methyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(2-hydroxyphenoxy)-1-{spiro[azepane-4,2'-chromene]-1-yl}ethan-1-one
1-[(2-chloro-4-fluorophenyl)methyl]-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
(3S,7S)-5-(2,5-dimethylfuran-3-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
2-amino-4-(1,3-dimethyl-1H-pyrazol-4-yl)-6-(furan-2-ylmethyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[(1S,2R)-2-aminocyclobutyl]-3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propanamide
3-(2-methoxyphenyl)-N-[2-(pyrimidin-2-ylmethyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]propanamide
methyl 2-[2-({4-[(3-chlorophenyl)methyl]piperazin-1-yl}methyl)phenoxy]acetate
2-cyclopropyl-5-[2-(3-fluorophenyl)azepane-1-carbonyl]pyrimidin-4-ol
[(4-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-2-yl}phenyl)methyl]dimethylamine
5-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N,N-dimethylpyridin-2-amine