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2-[(1-acetylpiperidin-4-yl)oxy]-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-methoxybenzamide
{2-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}urea
2-{4-[(5-methylthiophen-2-yl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
3-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-3,9-diazaspiro[5.6]dodecan-10-one
1-(4-{[(3R,4R)-3-hydroxy-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
(3aR,6aS)-2-{[3-(cyclopentyloxy)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole
1-(3-chloro-2-propoxyphenyl)-3-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]urea
1-(azocan-1-yl)-3-[2-methoxy-4-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-[(4-chlorophenyl)methyl]-4-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazine
N-[(1S,2R)-2-aminocyclobutyl]-1-benzoxepine-4-carboxamide
N-benzyl-5-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[(2-methyl-5-sulfamoylphenyl)formamido]-N-(1,3-thiazol-2-yl)acetamide
1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl})amine
1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(piperidin-1-yl)piperidine-4-carboxamide
(1S,4S)-N-[3-(4-hydroxypiperidin-1-yl)propyl]-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carboxamide
2-[methyl(2-phenylethyl)amino]-N-(oxan-2-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-3-(4-phenylbenzoyl)piperidine-1-carboxamide
3-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanamide
3-ethyl-5-{[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole
N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylpiperidine-3-carboxamide
methyl 4-{[(4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}phenyl)formamido]methyl}benzoate
3-(azocan-1-yl)-N-[(3S)-2-oxoazepan-3-yl]propanamide
1-(5-chloropyridin-2-yl)-4-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperazine
3,7-dimethyl-11-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,7,11-triazaspiro[5.6]dodecane
(2S,4R)-4-amino-N-ethyl-1-(2,2,6,6-tetramethylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-(2,2-dimethyloxan-4-yl)-N'-(3,5-dimethylphenyl)-N-ethylpropanediamide
methyl 5-oxo-5-[3-(4-phenylbenzoyl)piperidin-1-yl]pentanoate
6-ethoxy-4-methyl-2-(4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepan-1-yl)quinazoline
N-(1-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-4-[(quinoxalin-2-yl)amino]pyrrolidin-2-one
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-2-methoxypyridine-4-carboxamide
(3S,4S)-3-hydroxy-4-{methyl[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amino}-1λ6-thiolane-1,1-dione
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[3-(methylsulfanyl)propyl]propanamide
(4aR,8aS)-6-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-[(5-methylfuran-2-yl)methyl]-3-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-3-yl}propanamide
1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(pyrazin-2-yl)propan-1-one
8-chloro-2-({[1-(pyrazin-2-yl)propan-2-yl]amino}methyl)quinolin-4-ol
N-[(3-methyloxetan-3-yl)methyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]ethan-1-one
N-[(2-butyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-4-oxo-4H-chromene-2-carboxamide
N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)but-3-enamide
3-(4-methylphenyl)-5-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propyl}-1,2,4-oxadiazole
1-methyl-N-[2-(pyridin-2-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
1-cyclobutanecarbonyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)piperidine-4-carboxamide
N'-methyl-N'-phenyl-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]ethanediamide
1-(3-cyanophenyl)-3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-ethylurea
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1-propylpiperidin-4-amine
1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
4-[5-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)-1H-pyrazol-3-yl]phenol