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N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
3-[1-(3-fluoro-4-methoxybenzoyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
2-{[2-(dimethyl-1,3-thiazol-2-yl)ethyl]amino}-N-phenylbutanamide
N-benzyl-3-[({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)methyl]-N-methylimidazo[1,2-a]pyridine-2-carboxamide
1-(3,3-diphenylpiperidin-1-yl)-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
2-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-5-methoxy-4H-pyran-4-one
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-N'-(2,4,6-trimethylphenyl)butanediamide
4-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-3,4-dihydro-2H-1,4-benzothiazin-3-one
1-[1-(tert-butylcarbamoyl)propyl]-3-(2-ethoxyethyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(2,3-dimethoxyphenyl)ethyl]acetamide
3-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(propan-2-yl)phenyl]urea
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
methyl 4-({1-[(3,3-diphenylpropyl)carbamoyl]-6-azaspiro[2.5]octan-6-yl}methyl)benzoate
1-(4-methyl-1H-imidazole-5-carbonyl)-4-[(3-methylphenyl)methyl]piperazine
N-cyclohexyl-3-[(5,6-dimethylpyrimidin-4-yl)amino]propanamide
1-{2-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-oxoethyl}piperidin-2-one
methyl 1-[(3S,5S)-1-cyclopentyl-5-{[2-(1H-indol-3-yl)ethyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-({3-[(E)-2-phenylethenyl]phenyl}methyl)acetamide
2-{[(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]pyrrolidin-1-yl]methyl}-6-ethoxyphenol
1-({1-[(2-chloro-6-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]quinolin-8-ol
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-cyclopropyl-4-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]pyrrolidin-2-one
methyl (2S)-1-({4-[(2,4-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)pyrrolidine-2-carboxylate
6-cyclopentyl-N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-({[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}methyl)phenol
2-ethyl-8-(8-hydroxyquinoline-7-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{4-[2-(azepane-1-carbonyl)phenoxy]piperidin-1-yl}-2-methoxyethan-1-one
3-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
2-(1-benzothiophen-2-ylmethyl)-4-[4-(pyrazine-2-carbonyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-(pyridin-2-ylmethyl)-3-[(pyrimidin-4-ylmethyl)sulfamoyl]benzamide
4-benzyl-1-[(3,4-difluorophenyl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3,4-dimethyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-5-sulfamoylbenzamide
3-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-3-yl]-N-[(2,4-dimethoxyphenyl)methyl]propanamide
2-[6-chloro-3-(pyrrolidin-1-ylmethyl)imidazo[1,2-a]pyridine-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopropanecarboxamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidine
2-(2,3-dimethoxy-5-methylphenyl)-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridine
N-cyclohexyl-N-[2-(3,4-dimethoxyphenyl)ethyl]-1-methyl-1H-pyrazole-5-carboxamide
2-[4-(4-cyclohexylpiperazine-1-carbonyl)piperidin-1-yl]-6-ethoxy-4-methylquinazoline
1-[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl]-4-methylpiperazine
{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
6-[({[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}amino)methyl]-1,4-oxazepan-6-ol
1-(7-{[3-(dimethylamino)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)hexan-1-one
7-(2-propoxypropanoyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(3-methoxypropyl)-9-(3-phenyl-1,2,4-oxadiazol-5-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-[methyl(2-phenylethyl)amino]-N-[(2S)-pyrrolidin-2-ylmethyl]-2,3-dihydro-1H-indene-2-carboxamide
4-[(3-fluorophenyl)methyl]-3-{2-[4-(2-methylphenoxy)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-{2-[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridine-3-carboxamide