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5-{2-[2-(4-chloro-1-methyl-1H-indazol-3-yl)-1H-imidazol-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-({7-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazole
N-cyclopentyl-1-methyl-3-(2-methylpropyl)-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-5-carboxamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
3-[(4-ethylpiperazin-1-yl)methyl]-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-amino-6-(2-fluoro-4-hydroxyphenyl)-4-[2-(methoxymethyl)pyrimidin-5-yl]pyridine-3-carbonitrile
3-methyl-4-[1-(5-phenyl-1,2-oxazole-3-carbonyl)pyrrolidin-2-yl]-1,2,5-oxadiazole
2-(2-chloro-4-fluorophenoxymethyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
4-{[2-(1H-imidazol-2-yl)phenyl]formamido}-N-methylbutanamide
N-({4-[benzyl(ethyl)amino]quinazolin-2-yl}methyl)spiro[2.4]heptane-1-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
5-[(4-benzylpiperidin-1-yl)methyl]-N-[2-(1H-imidazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[2-(1H-indol-3-yl)ethyl]acetamide
N-{1-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
3-(1-{2-chloro-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-3-yl)-N-cyclopropylpropanamide
4-[(dimethylamino)methyl]-1-[(1-ethyl-1H-indol-4-yl)methyl]azepan-4-ol
N-[2-(2-ethylphenoxy)ethyl]-3-ethynyl-N-methylbenzamide
1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-(propan-2-ylsulfanyl)ethan-1-one
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-methanesulfonyl-1,4-diazepane
N-[1-(3-fluorophenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]oxolane-2-carboxamide
3-[4-(pyridin-2-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyridin-1-ium-1-olate
N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(propan-2-yloxy)ethyl]acetamide
1-(4-fluorophenyl)-3-methyl-5-[1-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazole
3-({[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)propane-1,2-diol
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(propan-2-yloxy)benzamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-(oxan-2-ylmethyl)-3-[(thiophen-2-ylmethyl)amino]benzamide
1-(2-{4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)piperazine
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]pyrrolidin-2-one
4-{1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}benzoic acid
2-[(4-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}piperidin-1-yl)methyl]pyridine
N-(2-ethoxyphenyl)-4-[(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-1-carboxamide
N-({2-[(dimethylamino)methyl]phenyl}methyl)-6-ethylpyrimidin-4-amine
1-[(6-methylpyridin-2-yl)methyl]-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1-(piperidin-1-yl)cyclohexane-1-carboxamide
(2S,4S)-4-amino-1-(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-N-methylpyrrolidine-2-carboxamide
3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
1-methyl-2-(1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-imidazol-2-yl)-1H-imidazole
methyl 4-(5-{[(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
1-(cyclopropylmethyl)-4-(3-fluoro-4-methoxyphenyl)-1H-pyrazole
4-methoxy-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]benzamide
1,2-dimethyl-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazine
3-{2-[(2S)-4-methyl-2-(propan-2-yl)piperazin-1-yl]-2-oxoethyl}-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
ethyl 5-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
2-methyl-4-(3-{1-[(1-methyl-1H-imidazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)-5-propylpyrimidine
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(oxan-4-yl)ethyl]acetamide
2-(3-methylbutyl)-8-(pyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-methyl-N-[2-methyl-1-(morpholin-4-yl)propan-2-yl]-1H-indole-3-carboxamide