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(2R,6S)-4-[1-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]-2,6-dimethylmorpholine
N-(2-{1-[(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}ethyl)pyrrolidine-1-carboxamide
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
2-[4-(3-methoxypyridin-2-yl)-1H-pyrazol-1-yl]-N-(1-propyl-1H-indazol-3-yl)acetamide
1-methyl-3-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-1-[1-(4-methylpyridin-2-yl)propan-2-yl]urea
5-{[benzyl(methyl)amino]methyl}-N-(3-hydroxy-2,2-dimethylpropyl)-1,2-oxazole-3-carboxamide
methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-N-[(5-methylfuran-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
5-(2,4-dimethoxyphenyl)-N-(oxolan-2-ylmethyl)-1,2,4-triazin-3-amine
4-{1-[(2,5-dimethoxyphenyl)methyl]piperidin-4-yl}-5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidine
(3aS,7aR)-2-[2-(5-fluoro-2-methyl-1H-indol-3-yl)acetyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
5-[2-(benzylamino)ethyl]-1-[(5-methylfuran-2-yl)methyl]pyrrolidin-2-one
N-[(2R,3R)-1'-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
2-(1-{[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carbonyl)pyridine
4-{6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
2-[1-(1,3-thiazol-2-yl)ethyl]-4-(4-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}piperidin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[(1R,3R)-3-aminocyclopentyl]-2-(ethylamino)pyrimidine-5-carboxamide
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-2-{3-[2-(trifluoromethyl)phenyl]-1H-pyrazol-1-yl}acetamide
4-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
methyl (2S)-2-[(1-{4-[(benzylcarbamoyl)methyl]phenyl}piperidin-4-yl)amino]-3-phenylpropanoate
N-cyclopropyl-N-{[4-(methylsulfanyl)phenyl]methyl}-1H-pyrazole-3-carboxamide
1-ethyl-4-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
N,N-dimethyl-6-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]pyrimidin-4-amine
1-(6,7-dimethoxy-4-methylquinolin-2-yl)-N-ethylpyrrolidine-3-carboxamide
2-[(1,4-dioxan-2-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3-(3-methyl-1H-pyrazol-1-yl)-1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
[(3S,5R)-1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
ethyl 5-(2-methyl-1,3-thiazole-4-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-methyl-2-oxo-8-(quinoline-4-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(cyclohex-1-en-1-yl)-1-{4-[5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
2-{4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-methyl-2-(5-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}furan-2-yl)-1H-1,3-benzodiazole
2-(1H-1,3-benzodiazol-1-yl)-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]propanamide
N-cyclopropyl-N-{[2-(4-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-2-(trifluoromethyl)benzamide
2-(3-cyclopropanecarbonyl-1H-indol-1-yl)-N-[(5-methylpyrazin-2-yl)methyl]acetamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
1-[(2S,4R)-4-(1H-1,2,3,4-tetrazol-1-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carbonyl]azepane
1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-4-(propan-2-yl)pyrimidin-2-amine
N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}-1H-1,2,3-triazole-5-carboxamide
N-ethyl-6-(quinolin-6-yl)pyridine-3-carboxamide
1-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
1-{7,7-dimethyl-5-[(pyrazin-2-yl)amino]-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-ol
N'-(2-tert-butylphenyl)-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]butanediamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-methanesulfonyl-N-methylpyrrolidine-2-carboxamide
8-[(4-methylphenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-benzyl-N-methyl-1-[(2,4,5-trimethoxyphenyl)methyl]piperidin-3-amine
3-(3,4-dimethoxyphenyl)-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpropanamide
5-butyl-1'-(quinolin-4-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]