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2-[4-(3-oxo-3,4-dihydroquinoxaline-2-carbonyl)morpholin-3-yl]acetic acid
7-{3-[(1R,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]pyridin-2-yl}-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-3-[(4-methoxy-2,5-dimethylphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[(3R,4S)-1-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-hydroxyacetamide
2-{3-[(3-chlorophenyl)methyl]-5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)morpholine-2-carboxamide
3-[2-(4-benzylpiperidin-1-yl)-2-oxoethyl]-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
N-[3-(1H-imidazol-1-yl)propyl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
1-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3-{1-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(6-chloropyridin-3-yl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
(1S,5R)-3-(3-chlorobenzenesulfonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(2,4-difluorophenyl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
2-{1,3-dimethyl-4-[3-(propoxymethyl)pyrrolidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-(1,3-thiazole-4-carbonyl)piperidine-4-carboxylic acid
1-[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-3-(4-phenylphenyl)propan-1-one
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(2,6-difluorophenyl)ethan-1-one
5-[(3-fluorophenyl)methyl]-5-[1-(furan-3-ylmethyl)piperidin-4-yl]-3-(2-methylpropyl)imidazolidine-2,4-dione
ethyl 3-[(4-fluorophenyl)methyl]-1-(5-methylthiophene-2-carbonyl)piperidine-3-carboxylate
2-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-6-fluoroquinoline
(2S,4S)-4-amino-1-[3-(4-methylphenyl)-1-phenyl-1H-pyrazole-4-carbonyl]pyrrolidine-2-carboxylic acid
3-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-[4-(furan-2-yl)butan-2-yl]urea
(1-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-3-(prop-2-en-1-yl)piperidin-3-yl)methanol
4-(but-2-ynoyl)-6-[(4-fluorophenyl)methoxy]-1-(propan-2-yl)-1,4-diazepan-2-one
ethyl 2-(1-{2-[(2-fluorophenyl)methyl]-1,3-benzoxazole-6-carbonyl}piperidin-2-yl)acetate
7-(2-oxo-1,3-oxazolidin-3-yl)-4-[(1s,4s)-4-aminocyclohexyl]-1,2,3,4-tetrahydroquinolin-2-one
3-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-6-methyl-1H-indole
N-[2-(pyridin-2-yl)ethyl]-3-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(pyridin-3-ylmethyl)amine
2-(1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)-4-methyl-1H-1,3-benzodiazole
3-(5-{[4-(2-oxoimidazolidin-1-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
1-[(5-acetylthiophen-3-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
3-(3-methoxyphenyl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
2-methyl-N-[1-(7-{[3-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-3-carboxamide
1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
2-[5-methyl-4-(4-propylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(thiophen-2-yl)pyrimidine
4-[1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)pyrrolidin-2-yl]-3,5-dimethyl-1,2-oxazole
(4aR,7aS)-1-cyclobutanecarbonyl-4-(3,5-dimethylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2,3-dimethoxyphenyl)-2-(3-oxopiperazin-1-yl)acetic acid
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(ethanesulfinyl)ethyl]-3-(2-methylpropyl)-1H-1,2,4-triazole
5-{2-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-(pyrazin-2-yl)-N4-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-{2-[(4-cyano-4-methylpiperidin-1-yl)methyl]-4-(thiophen-3-yl)phenoxy}acetic acid
6-({2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-[3-cyclopentyl-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]-3,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[(2-chloropyridin-3-yl)methyl]-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methylbenzamide
1-(4-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(1H-indol-3-yl)ethan-1-one