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(2S,4S)-N-ethyl-1-(1H-imidazol-4-ylmethyl)-4-(3-phenylpropanamido)pyrrolidine-2-carboxamide
2-[(3-propylmorpholin-4-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
1-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(pyridin-3-yl)ethan-1-one
4-[1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]piperazine-1-sulfonamide
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-5,6-dimethylpyridine-3-carboxamide
1-{4-[(2,3-dihydroxypropyl)(methyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N,N-dimethyl-3-[1-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)piperidin-3-yl]propanamide
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)({[2-(furan-2-yl)pyrimidin-5-yl]methyl})methylamine
1-(methoxymethyl)-N-{2-[2-(trifluoromethyl)phenyl]ethyl}cyclobutane-1-carboxamide
1-[4-({4-[(2,3,6-trifluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydroisoquinolin-1-one
N-methyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-(propan-2-yl)acetamide
methyl 2-{[(3-chlorophenyl)methyl]sulfamoyl}-6-(1-methylcyclopropanecarbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N3-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-N5-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-[(3-chloro-4-fluorophenyl)methyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
1-(4-{[2-(2,3-dimethoxyphenyl)ethyl]amino}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(4-methyl-1H-imidazole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N3,N3-diethyl-N1-[2-methyl-3-(pyrrolidin-1-yl)phenyl]piperidine-1,3-dicarboxamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-ethyl-1,2-oxazole-3-carboxamide
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(1,3-dihydroxypropan-2-yl)-decahydro-1,6-naphthyridin-2-one
3-methyl-1-{1-[6-(pyridin-4-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
N-methyl-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole
2-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-5-methoxy-4H-pyran-4-one
5-acetyl-N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)thiophene-3-carboxamide
N-{2-[2-(1H-imidazol-1-yl)propanamido]-4-methylphenyl}cyclohexanecarboxamide
N-[1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-4-phenylbutanamide
4-(1H-imidazol-2-yl)-1-[5-(4-methoxyphenyl)furan-2-carbonyl]piperidine
3-methyl-1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazine
4-(1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-imidazol-2-yl)-2,1,3-benzoxadiazole
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
4-{[3-(2-chlorophenoxy)azetidin-1-yl]methyl}-5-cyclopropyl-1-methyl-1H-pyrazole
9-(2-methyl-5-propylpyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(2-chlorophenyl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]furan-2-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}propanamide
1-methyl-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)propan-1-one
3-ethyl-1-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
3-[2-(2,4-difluorophenyl)ethyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine
3-ethyl-1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-3-ol
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(cyclopropylmethyl)-N-propylacetamide
methyl 3-(furan-2-amido)-1-methyl-5-[(3-methylbutyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[(1-methyl-1H-pyrrol-2-yl)methyl]-N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]piperidine-4-carboxamide
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-N-methylacetamide
2,2-dimethyl-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)oxane-4-carboxamide
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-3-(1H-pyrazol-1-yl)butanamide
4-methyl-1-[(3-phenyloxolan-3-yl)methyl]piperidine-4-carbonitrile
(4aR,7aS)-1-(2-methoxyethyl)-4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione