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2-(dimethylamino)-2-(3-fluorophenyl)-1-[3-(pyridin-2-yl)azetidin-1-yl]ethan-1-one
1-(4-{[2-(4-fluorophenoxy)ethyl]amino}-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
N-[2-(1H-indol-3-yl)ethyl]-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
3-{3-[({[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}amino)methyl]-1H-indol-1-yl}propanamide
3-hydroxy-3-{[3-(hydroxymethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-(2-methoxyethyl)piperidin-2-one
5-(2-methoxyacetamido)-N,1-dimethyl-N-(oxan-2-ylmethyl)-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
2-(3-chlorophenyl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
[(3-{[1-(2,2-dimethyloxane-4-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](1H-imidazol-2-ylmethyl)methylamine
[9-(2-cyclopropylpyrimidine-5-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
1-(2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-2-methyl-1H-indole-3-carbonitrile
N-({5-[(3-cyanophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
2-(2-chloro-4-fluorophenyl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
3-{[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
2-[4-(1,3-benzothiazol-2-ylmethyl)-1-methylpiperazin-2-yl]ethan-1-ol
N-{1-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methylpyridine-2-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]benzamide
2-[2-ethoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
4'-(3,3-dimethylbutyl)-1-(2-methylpropyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(3R)-1-[(1-{[1-(thiophene-3-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-3-ol
3-({1-[2-(azepan-1-yl)acetyl]pyrrolidin-3-yl}methyl)benzamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)-1H-imidazole
4-cyano-N-[(2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)benzamide
N-ethyl-N-(oxolan-2-ylmethyl)-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(2,2-dimethylpropanoyl)-N-[2-(pyridin-2-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-[({[4-(3-fluorophenyl)oxan-4-yl]methyl}carbamoyl)amino]-4-methylbenzamide
2-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}quinolin-4-ol
N-(2-hydroxyethyl)-1-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
1-ethyl-N-[3-(2-fluorophenyl)propyl]-5-oxopyrrolidine-3-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
methyl 3-{[(9-methyl-9H-carbazol-3-yl)formamido]methyl}-5-[2-(1H-pyrazol-1-yl)acetamido]benzoate
2-methyl-9-{[3-(trifluoromethyl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(1R,7S)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-(3-methylbutyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-(4-{[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
N-[5-(3-phenylpiperidine-1-carbonyl)-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazol-7-yl]acetamide
(1R,3S)-3-(2-aminoethoxy)-7-[(4-ethoxyphenyl)methyl]-7-azaspiro[3.5]nonan-1-ol
5-[1-(2-ethylbutanoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-{2-[7-(1-benzofuran-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclobutanecarboxamide
2-(azepan-1-yl)-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
(1S,5R)-N-(2H-1,3-benzodioxol-5-yl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
6-[3-(2,5-difluorobenzoyl)piperidin-1-yl]-N-ethyl-N-methylpyrimidin-4-amine
9-(1,3-dimethyl-1H-indole-2-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-cyclopentyl-N-({4-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[2-(2-fluorophenyl)ethyl]-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
methyl 6-[2-(cyclohexylmethyl)morpholine-4-carbonyl]pyridine-3-carboxylate
1-[(3-methoxyphenyl)methyl]-N-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidin-3-amine
1-[(3-fluorophenyl)methyl]-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-1,4-diazepane
N-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-cyclobutylacetamide
4-{2,2-dimethyl-3-[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]propyl}morpholine