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1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-4-(6-methylpyridin-2-yl)piperazine
(1-{2-amino-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3-(prop-2-en-1-yl)piperidin-3-yl)methanol
3-({[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
1-(pyridin-2-ylmethyl)-4-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1,4-diazepane
1-methoxy-8-[2-(7-methyl-2-oxo-2H-chromen-4-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-[2-methyl-4-oxo-1-(oxolan-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
N-[2-(2-methyl-1H-indol-3-yl)ethyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
3-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-ol
1-(2,2-dimethyloxane-4-carbonyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
5-chloro-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]pyridine
4-(3-methylphenoxy)-1-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylic acid
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-methyl-2-[4-(piperidine-1-carbonyl)morpholin-3-yl]acetamide
2-(3-chloro-4-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
1-[(4-chlorophenyl)methyl]-N-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
5-ethyl-2-(3-{1-[(3-methylpyridin-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
1-(3-methanesulfonamido-4-methoxyphenyl)-3-[1-(3-methylphenyl)cyclopropyl]urea
2-methyl-5-(propan-2-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
7-(2-hydroxyethyl)-2-{6-methylthieno[2,3-d]pyrimidin-4-yl}-2,7-diazaspiro[4.5]decan-6-one
ethyl 3-({5-cyclopropyl-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazol-4-yl}formamido)propanoate
methyl 5-{[1-(3,4-dimethoxyphenyl)propan-2-yl]amino}-3-acetamido-1-ethyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
3-(2-hydroxyphenyl)-N-[3-(methylsulfanyl)propyl]-1H-pyrazole-5-carboxamide
2-amino-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-6-(propan-2-yl)pyrimidine-4-carboxamide
1-ethyl-3-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
4-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]-2,6-dimethylpyrimidine
1-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
1-{[1-(1-methylpiperidin-4-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(pyridin-2-yl)ethyl]amine
[(3-{[1-(2,5-dimethoxybenzoyl)piperidin-4-yl]oxy}phenyl)methyl](1H-imidazol-2-ylmethyl)methylamine
1-[1-(hydroxymethyl)-9-(3-methylbutyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-(1,3-thiazol-5-yl)ethan-1-one
8-(2,2-dimethylpropyl)-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-({[(3R,4R)-1-(2,3-dihydro-1H-indene-5-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
N-cyclopropyl-1-[1-(2,5-dimethylpyrimidin-4-yl)piperidin-4-yl]piperidine-3-carboxamide
4-[1-(oxane-4-carbonyl)pyrrolidin-3-yl]benzoic acid
4-(6-methyl-9H-purin-9-yl)benzamide
(4S)-4-(methoxymethyl)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3,3-dimethylpiperidin-4-ol
1-(2H-1,3-benzodioxole-5-carbonyl)-N-(4-fluorophenyl)piperazine-2-carboxamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
5-[2-(pyridin-2-yl)-1H-imidazol-1-yl]pyridin-2-amine
N-{1-[1-(1H-indole-2-carbonyl)piperidin-4-yl]-2-phenylethyl}-N,2-dimethylpropanamide
1-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl){[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amine
(3S,4S)-1-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N-cyclopropyl-3-{4-[(dimethylcarbamoyl)methyl]phenyl}benzamide
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[5-(morpholin-4-yl)pentyl]acetamide
(1H-imidazol-4-ylmethyl)(2-methylpropyl)[(3-methylthiophen-2-yl)methyl]amine
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2,6,8-trimethylquinoline-4-carboxamide
1-ethyl-5-(1H-imidazol-2-ylmethyl)-N-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide