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N-[(2S,4R,6S)-2-(2,1,3-benzothiadiazol-4-yl)-6-ethyloxan-4-yl]benzamide
N-({2-[(dimethylamino)methyl]phenyl}methyl)-N-methylfuran-3-carboxamide
3-ethyl-2-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-1H-indole
2-methyl-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-1H-1,3-benzodiazole-5-carboxamide
ethyl 1-(1H-1,3-benzodiazol-2-ylmethyl)-3-benzylpiperidine-3-carboxylate
1-[3-({7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)phenyl]ethan-1-one
5-(4-carbamoylphenyl)-2-chloro-N-methylbenzamide
6-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]-2-(2-methoxyethyl)-1,3-benzoxazole
3-(2-fluorophenyl)-N-methyl-N-[2-(morpholin-4-yl)ethyl]-3-phenylpropanamide
1-[(6-methoxypyridin-3-yl)methyl]-N,N-dimethylazepan-4-amine
N-methyl-N-[2-(2-methylphenyl)-1-{1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidin-4-yl}ethyl]-2-(1H-pyrazol-1-yl)acetamide
8-[2-(aminomethyl)-5-chloro-2,3-dihydro-1-benzofuran-7-yl]-2-methylquinolin-4-ol
[(3R,4R)-1-(1H-indole-6-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-propyl-1,3-thiazole-4-carboxamide
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(oxan-4-yl)ethyl]acetamide
2-[1-cyclopropyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]spiro[2.4]heptane-1-carboxamide
3-methyl-8-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-chloro-2,5-dimethyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}benzene-1-sulfonamide
N-[(2R,3R)-1'-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-(2-hydroxyethyl)-5-[3-(1H-indol-3-yl)propanoyl]-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
4-[(2-chlorophenyl)methyl]-1-[(4-fluoro-3-methoxyphenyl)methyl]-1,4-diazepan-5-one
4-methyl-6-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]pyrimidin-2-amine
1-(2-chlorophenyl)-4-(1H-indazole-3-carbonyl)-5-methylpiperazin-2-one
2-(benzyloxy)-N-[(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)methyl]acetamide
1-(1,3-benzothiazol-2-yl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-4-amine
3-[(2,3-dimethoxyphenyl)methyl]-5-[1-(2-ethylbutyl)piperidin-4-yl]-5-methylimidazolidine-2,4-dione
1-(dimethylamino)-2-{4-[(4-methoxynaphthalen-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
(1R,3S)-7-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
4-ethyl-3-{1-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
1-[(1S,3R)-1-[2-(dimethylamino)ethoxy]-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
N,N-dimethyl-2-[(1S,5R)-6-[4-(methylsulfanyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
7-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-7-propyl-2,7-diazaspiro[4.5]decan-6-one
7-(3,4-dimethoxyphenyl)-9-methoxy-4-(propan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(1-{3-[(dimethylamino)methyl]-1,2,4-oxadiazol-5-yl}cyclohexyl)-3,4-dimethylaniline
N-[2-(4-methylmorpholin-2-yl)ethyl]-2-propylpyridine-4-carboxamide
(3-{[5-(1H-1,3-benzodiazol-6-yl)pyridin-2-yl]oxy}propyl)dimethylamine
N-(butan-2-yl)-2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzamide
1-(4-{3-[2-(2-hydroxyphenyl)ethyl]-4H-1,2,4-triazol-4-yl}phenyl)ethan-1-one
6-{[3-(2-ethyl-1H-imidazol-1-yl)propyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
6-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,6-dihydropyridine-3-carboxamide
4-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}morpholine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4H-thieno[3,2-b]pyrrole-5-carboxamide
3-{1-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-1H-imidazol-2-yl}phenol
2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]acetic acid