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2-[(4-methoxyphenyl)methyl]-4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}morpholine
3-[2-(4-cyclopentylpiperazin-1-yl)-2-oxoethyl]-3-(2-methylphenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
[(3-fluorophenyl)methyl](2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
N-[(4-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethoxy}-3-methoxyphenyl)methyl]-N-[(3S)-2-oxoazepan-3-yl]cyclopropanecarboxamide
methyl 9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-3-[(2,4,5-trimethylphenyl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
6-{3-hydroxy-5-[2-(piperidin-2-yl)ethyl]phenyl}-N,N-dimethylpyrazine-2-carboxamide
2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]propanamide
(1S,3R)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-[(pyrrolidine-1-sulfonyl)amino]cyclopentane-1-carboxamide
N-cyclopropyl-3-({1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
4-(3-methylphenoxy)-1-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidine
4-(2,6-dimethylpyridin-3-yl)-N-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-2-amine
2-[(5-{1-[(5-methylpyrazin-2-yl)methyl]-1H-imidazol-2-yl}pyrimidin-2-yl)amino]acetic acid
1-[7-(3-chlorophenyl)-9-(thiophen-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
3-(2-methoxyethyl)-1-{thieno[3,2-d]pyrimidin-4-yl}piperidine-3-carboxylic acid
1-(3-hydroxyphenyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxamide
4-[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]thiomorpholine
{4-[(4-methoxyphenyl)methyl]-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl}methanol
2-(morpholine-4-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
3-ethyl-N-[(2S)-1-methoxy-3-phenylpropan-2-yl]-1,2-oxazole-5-carboxamide
methyl 4-({4-[4-(2-methylpropyl)-2,5-dioxo-1-[2-(thiophen-2-yl)ethyl]imidazolidin-4-yl]piperidin-1-yl}methyl)benzoate
3-(1-methyl-1H-pyrrol-2-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
5-(3,3-diphenylpiperidine-1-carbonyl)piperidin-2-one
4-{[(5-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}pyridine
6-[4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-5-(methoxymethyl)furan-2-carboxamide
N-(butan-2-yl)-2-(pyridin-3-yloxy)-N-(pyridin-4-ylmethyl)acetamide
8-(5-fluoropyridine-3-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}dimethylamine
N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-[2-(dimethylamino)ethyl]-N-{[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl}-2-(3-methyl-1H-pyrazol-1-yl)acetamide
1-ethyl-8-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-3-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-N-[(3-methylquinoxalin-2-yl)methyl]oxan-4-amine
(3R,4R)-4-cyclobutyl-3-methyl-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-4-ol
2-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-N-methyl-1,3-benzoxazole-6-carboxamide
1-methyl-4-phenyl-3-{[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(3aR,5R,6S,7aS)-2-(6-amino-2-methylpyrimidin-4-yl)-octahydro-1H-isoindole-5,6-diol
N-[(7-{[3-(furan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-3-(pyridin-3-yl)propanamide
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(6-methyl-2-propylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
8-(isoquinolin-1-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(4-acetyl-1,4-diazepan-1-yl)-2-(2-fluoro-4-methylphenyl)acetic acid
5-{3-[1-(dimethylamino)ethyl]phenyl}-2,3-difluorophenol
methyl 2-(1H-pyrazol-3-yl)pyridine-4-carboxylate
2-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1,2-oxazolidine
1-methyl-3-(2-phenylethyl)-8-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4R)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-1-[(4-fluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
N-{3-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-oxopropyl}acetamide
N-(1H-1,2,3-benzotriazol-4-yl)-2-butyl-4-methyl-3-oxopiperazine-1-carboxamide
1-{2-[3-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one