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1-methyl-N-[2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-1H-pyrazole-5-carboxamide
ethyl 2-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]acetate
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(2,6-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-6-ethylpyrimidin-4-amine
ethyl 3,5-dimethyl-4-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]-1H-pyrrole-2-carboxylate
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]benzamide
({3-methoxy-2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)(morpholin-2-ylmethyl)amine
4-(2-amino-6-methylpyrimidin-4-yl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-(2-fluorophenyl)-N-[3-(1H-imidazol-1-yl)butyl]pyrazolo[1,5-a]pyrimidin-7-amine
8-(oxolane-3-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N,N-dimethyl-3-[({2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}amino)methyl]pyridin-2-amine
1-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-3-(1,1-dioxo-1λ6-thiolan-3-yl)urea
1-[(3-methylpyridin-2-yl)methyl]-4-[3-(trifluoromethyl)benzoyl]piperazine
4-{[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]methyl}-1-ethyl-1H-pyrrole-2-carbonitrile
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-8-methoxy-4-methylquinoline
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[1-(6-methylpyridine-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
6,7-dimethoxy-3-{[methyl(2-methylpropyl)amino]methyl}-1,2-dihydroquinolin-2-one
4-[3-(benzyloxy)piperidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
N-ethyl-6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridazin-3-amine
1-{4-[1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]phenyl}-3-(oxolan-3-ylmethyl)urea
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-methoxy-N-methylpyridine-3-carboxamide
4-(2-methoxyethoxy)-1-(1H-pyrazole-3-carbonyl)piperidine
N-[(4-methylphenyl)methyl]-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
1-(4-{[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2,2-dimethylbutan-1-one
dimethyl(2-{2-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)propanamide
2-(morpholin-3-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-[(1S)-1-carbamoyl-3-methylbutyl]-N'-cyclooctylbutanediamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)propanamide
[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]{[4-(pyrimidin-2-yloxy)phenyl]methyl}amine
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}acetamide
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
1-tert-butyl-5-{[(cyclopropylmethyl)sulfanyl]methyl}-3-methyl-1H-1,2,4-triazole
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-methyl-N-(1,2-oxazol-3-ylmethyl)pyridin-2-amine
2-{1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-3-yl}benzoic acid
2-[(2-amino-6-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidin-4-yl)amino]ethan-1-ol
1-({5-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]furan-2-yl}methyl)-1H-pyrazole
4-benzyl-3-[1-(6-methoxypyrimidin-4-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(1,3-thiazol-2-yl)ethyl]piperidine-3-carboxamide
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]ethan-1-one
3-(1-benzyl-1H-pyrazol-5-yl)-1-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}urea
6-methyl-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carboxamide
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-(oxolan-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(4-{1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
3-[(3S,4R)-4-amino-3-methoxypiperidine-1-carbonyl]-6-ethyl-1,5-dimethyl-1,2-dihydropyridin-2-one
1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
2-{1-[(2-fluorophenyl)methyl]-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
3-{3-[(3,4-dimethoxyphenyl)amino]piperidine-1-carbonyl}-1-methyl-1,4-dihydroquinolin-4-one
3-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile