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N-[2-(3-fluorophenyl)ethyl]-5-{4-hydroxy-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1-benzofuran-2-carboxamide
(2S,4S,5R)-5-(2-fluorophenyl)-4-(3-hydroxyazetidine-1-carbonyl)-1-methylpyrrolidine-2-carboxylic acid
5-ethyl-5-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
1-(2,3-dimethylphenyl)-4-[3-(pyrrolidin-1-yl)piperidin-1-yl]piperidine
6-cyclopentyl-1-methyl-4-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-1H-pyrazolo[3,4-d]pyrimidine
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[2-(pyridin-3-ylformamido)ethyl]acetamide
3-[1-(3-fluoro-4-methoxybenzoyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
(4aS,7aR)-1-[2-(3-methoxyphenoxy)acetyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[2-(pyridin-3-yl)pyrrolidin-1-yl]ethan-1-one
4-methyl-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1,2,5-oxadiazole-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}oxolane-2-carboxamide
4-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazin-2-one
2-(4-fluorophenyl)-1-(1,3-thiazol-4-ylmethyl)piperidine
4-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetyl}piperazine-1-sulfonamide
N-[(4-hydroxyazepan-4-yl)methyl]-2-methyl-1-benzofuran-7-carboxamide
1-(5-chloro-2-fluorobenzoyl)-N-phenylpiperidin-3-amine
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]acetamide
8-fluoro-N-[3-(1H-1,2,4-triazol-1-yl)propyl]quinoline-2-carboxamide
6-methoxy-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
(1R,5R)-3-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-(dimethyl-1H-1,2,4-triazol-3-yl)-2-methyl-4-(2-methylphenyl)piperazine-1-carboxamide
8-[3-(1H-indol-3-yl)propanoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-{1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-3-yl}-N,N-dimethylpropanamide
(3R,9R)-11-[(2-fluoro-5-methylphenyl)methyl]-5-thia-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
2-[2-(4-methoxypiperidin-1-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
4-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-1λ6-thiomorpholine-1,1-dione
ethyl 3-[(4-fluorophenyl)methyl]-1-propanoylpiperidine-3-carboxylate
N-[(2-chlorophenyl)methyl]-3-[1-(quinolin-8-ylmethyl)piperidin-3-yl]propanamide
2-ethyl-5-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)pyrimidine
{2-[8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-2-oxoethyl}urea
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-(1H-pyrazol-4-yl)pyridine
2-(4-chlorophenyl)-4-[(4-methoxypiperidin-1-yl)sulfonyl]morpholine
N-[(1-benzylpiperidin-4-yl)methyl]-1-cyclopropyl-1H-pyrrole-2-carboxamide
N-(4-{[(1H-indol-4-ylmethyl)carbamoyl]methyl}phenyl)butanamide
{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}(methyl)(quinolin-2-ylmethyl)amine
methyl 3-(2-chlorobenzamido)-5-[(2,2-dimethylpropanamido)methyl]benzoate
methyl 3-(2,4-dichloro-5-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxylate
(1S,5R)-3-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3,5-dimethyl-1-[1-(3-propyl-1H-pyrazole-5-carbonyl)azetidin-3-yl]-1H-pyrazole
5-(3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-3-oxopropyl)imidazolidine-2,4-dione
7-[2-(benzyloxy)ethyl]-2,7-diazaspiro[4.5]decane
N-cyclopropyl-3,5-dimethyl-N-[(5-methylthiophen-2-yl)methyl]-1H-indole-2-carboxamide
5-methyl-1-propyl-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
1-[4-({methyl[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amino}methyl)thiophen-2-yl]ethan-1-one
2-[1-(2H-1,3-benzodioxol-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-3-(piperidine-1-carbonyl)pyrazine
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[3-(2-methoxyphenyl)propyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
(2R,3R)-3-[(2-hydroxyethyl)(methyl)amino]-1'-(pyrazin-2-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(1R,2R)-2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}(propyl)amino)cyclohexan-1-ol