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N-[3-(3,4-dimethylphenoxy)propyl]-N-methyl-3-(3-methyl-1H-1,2,4-triazol-5-yl)propanamide
(3aS,6aS)-2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(1-cyclobutanecarbonylpiperidin-4-yl)-3-(pyrrolidine-1-carbonyl)piperidine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
5-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
4-{1-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]piperidin-3-yl}benzoic acid
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-indol-1-yl)ethyl]acetamide
2-[(3,4-dimethoxyphenyl)methyl]-4-{4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
2-({[(3R,4R)-1-[(3-chloro-4-methoxyphenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2,4-dimethyl-N-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]methyl}benzamide
N-[(1R,3S)-3-{[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]carbamoyl}cyclopentyl]pyrrolidine-1-carboxamide
N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-[(trimethylpyrazin-2-yl)methyl]piperidine-3-carboxamide
(1R,5R)-6-(2-methoxyethyl)-3-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
2-acetyl-8-{7-methylthieno[3,2-d]pyrimidin-4-yl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-2-methoxypyridine-3-carboxamide
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1-(pyridin-2-ylmethyl)urea
4-[(4-fluorophenyl)methyl]-1-(4-methylbenzoyl)-3-(propan-2-yl)-1,4-diazepan-5-one
(4aS,7aR)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-({3-azaspiro[5.5]undecan-9-yl}amino)-1-(pyridin-3-yl)ethan-1-ol
3-{[(3R)-3-methylpiperazin-1-yl]sulfonyl}-N-(oxan-4-ylmethyl)benzamide
3-[2-(dimethylamino)ethyl]-8-[(3-hydroxy-4-methoxyphenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2,1,3-benzoxadiazol-4-ylmethyl)-N,N-dimethylazepan-4-amine
N-({1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}methyl)-1,2,5-oxadiazole-3-carboxamide
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,4-diazepane
1-[2-butyl-4-(4-chlorophenyl)-5-oxopiperazine-1-carbonyl]cyclopropane-1-carboxamide
N,N-dimethyl-5-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)pyridin-2-amine
1-(cyclobutylmethyl)-4-(5-ethyl-1H-pyrrole-2-carbonyl)-1,4-diazepan-6-ol
2-(2-hydroxyethyl)-8-[(2-methoxy-4-methylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-{3-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,1,3-benzoxadiazol-1-ium-1-olate
2-[2-(pyridin-4-yl)-4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-amine
3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)pyridin-1-ium-1-olate
1-[2-(dimethylamino)ethyl]-4-ethyl-3-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{4-[(3,5-difluorophenyl)methyl]-1-[(2-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[(5-methylpyrazin-2-yl)methyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
5-(3,4-dimethylphenoxymethyl)-3-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1,2-oxazole
1-[(2E)-3-phenylprop-2-en-1-yl]-4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-1,2,3-triazole
4-cyclohexanecarbonyl-7-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3-phenyl-1,2-oxazole
N-(1-{7-[(3,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)furan-3-carboxamide
1-[3-({3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
N-[5-carbamoyl-2-(3-methylpiperidin-1-yl)phenyl]-5-chloro-6-oxo-1,6-dihydropyridine-3-carboxamide
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(pyridin-4-ylmethyl)amine
4-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}-N,5-dimethyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
3-(2-butoxyacetamido)-2-methyl-N-(1,3-thiazol-2-yl)benzamide
2-[2-(pyridin-4-yl)quinoline-4-carbonyl]-1,2-oxazolidin-4-ol
7-(2-methylphenyl)-4-(thiophene-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[4-(3-fluorophenyl)phenyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-amine
3-(4-chloro-1H-pyrazol-1-yl)-1-[2-(furan-2-yl)azepan-1-yl]propan-1-one
N-{[5-(3-phenylbutyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}methanesulfonamide
2-(2-fluoro-5-methoxyphenyl)-5-methyl-4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1,3-oxazole