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1-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-(furan-2-ylmethyl)-3-[5-(4-methylphenoxymethyl)-1,3,4-thiadiazol-2-yl]urea
1-[4-(furan-3-yl)phenyl]-2-(morpholin-4-yl)ethan-1-ol
2-(4-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}pyrimidin-5-yl)acetic acid
4-({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}sulfonyl)morpholine
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
6-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
5-methyl-N-[1-(pyridin-3-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
3-{[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl](pyridin-4-ylmethyl)amino}propan-1-ol
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-(3-phenylpropyl)pyrrolidin-2-one
3-{[4-({1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}amino)-6-methylpyrimidin-2-yl]amino}phenol
2-[(2-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)methyl]pyridine
N-cyclopentyl-4-[4-(piperazin-1-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
4-ethyl-3-({1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-(piperazin-1-yl)acetamide
4-chloro-5-{[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
N-(adamantan-2-yl)-6-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidin-3-amine
9-methoxy-4-(3-methoxybenzoyl)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2,6-dimethoxy-4-{1-[3-(pyridin-2-yl)propyl]-1H-imidazol-2-yl}phenol
2-amino-4-[3-(1H-pyrazol-1-yl)phenyl]-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
7-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-1,2-dihydroisoquinolin-1-one
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}imidazo[1,2-a]pyrimidine-2-carboxamide
(1S,5R)-6-(3-methyl-1H-pyrazole-5-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(2,4-dimethoxyphenyl)methyl]-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
1-(1H-indole-5-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
6-[(diethylamino)methyl]-N-(3,4-dimethylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-(2-fluorophenyl)-N-methyl-1H-pyrazole-5-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-(6-cyanopyridin-3-yl)-3-(1-methoxypropan-2-yl)urea
4-[2-(1-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]phenol
N-ethyl-2-[4-fluoro-3-(hydroxymethyl)phenyl]benzamide
(1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-yl)methanamine
1-(furan-2-yl)-2-{3-methyl-3,9-diazaspiro[5.6]dodecan-9-yl}ethane-1,2-dione
4,6-dimethyl-3-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
3-[5-(2-chloro-6-fluoro-3-methylphenyl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
2-(2,6-difluorophenyl)-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]acetic acid
2,5-dimethyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
ethyl 2-[1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)piperidin-2-yl]acetate
N-(2-methoxy-5-methylphenyl)-3-(3-methylthiophene-2-carbonyl)piperidine-1-carboxamide
N-[(3S,7S,8aS)-3-[(4-chlorophenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methoxybenzamide
3-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(methylsulfanyl)phenyl]urea
({2-[(2-chloroprop-2-en-1-yl)oxy]-6,7-dimethoxyquinolin-3-yl}methyl)[(2,3-difluorophenyl)methyl]amine
5-cyclopropanecarbonyl-1'-[(4-methyl-1H-imidazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1S,9S)-11-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N,N-dimethylbenzamide
N-[(2-fluorophenyl)methyl]-4-(4-{[2-(furan-2-yl)ethyl]amino}piperidin-1-yl)benzamide
1-(4-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)propan-1-ol
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-3-amine
2-({[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}amino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-{1-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}pyridine