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methyl({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
2-ethyl-9-[(3-hydroxyphenyl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(4-phenylbutan-2-yl)({2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
N-[3-(ethylcarbamoyl)-2-methylphenyl]-4-(1H-pyrrole-2-carbonyl)piperazine-1-carboxamide
N-{1-[1-(5-chloro-2-fluorobenzoyl)piperidin-4-yl]-2-phenylethyl}-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
4-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyridine
2-methoxy-5-{[1-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenol
5-(1-cyclopentyl-4-hydroxypiperidin-4-yl)-N-(3,4-dimethoxyphenyl)-1-benzofuran-2-carboxamide
N-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}oxolan-3-amine
(4aS,7aR)-1-(2-aminoacetyl)-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-tert-butyl-4-[({2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}(methyl)amino)methyl]pyrrolidin-2-one
3-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-2-methyl-6H,7H-pyrazolo[1,5-d][1,2,4]triazin-7-one
[1-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
ethyl 3-[(2-methylphenyl)methyl]-1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperidine-3-carboxylate
4-(1H-imidazol-4-yl)-6-methyl-2-oxo-N-{[3-(trifluoromethyl)phenyl]methyl}-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-ethyl-2-(2-fluoro-5-methoxyphenyl)benzamide
N-{3-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]phenyl}acetamide
3-(6-methoxynaphthalene-2-carbonyl)-1-(prop-2-ene-1-sulfonyl)piperidine
N-methyl-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]-N-[2-(pyridin-2-yl)ethyl]pyridin-2-amine
1-methyl-9-{thieno[2,3-d]pyrimidin-4-yl}-1,4,9-triazaspiro[5.5]undecan-5-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(1H-1,2,4-triazol-1-yl)benzamide
1-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-4-[(dimethylamino)methyl]azepan-4-ol
1-({1-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]cyclopropyl}methyl)-1H-pyrazole
2-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
(1S,6R)-9-(3-chloro-2-methylbenzenesulfonyl)-3,9-diazabicyclo[4.2.1]nonane
8-{3-[(diethylamino)methyl]-4-methoxyphenyl}-2H,5H,6H,7H,8H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-[2-(4-{[(2-ethylbutyl)(methyl)amino]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]methanesulfonamide
N-[(2-methylphenyl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
1-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-3-phenylprop-2-yn-1-one
2-(2-methyl-1H-imidazol-1-yl)-1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-{pyrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidin-3-amine
1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
3-benzyl-1-(3-methoxypropyl)-8-[(5-methylthiophen-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}acetamide
5-{5-[5-(oxolan-2-yl)thiophene-2-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-1,2-oxazole
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(pyridine-2-carbonyl)piperidin-3-yl]propan-1-ol
1-(3,6-dimethylpyrazin-2-yl)-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
4-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
1-[1,3-dioxo-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-[1-(furan-2-yl)ethyl]-N-methylpiperidine-4-carboxamide
N-[2-(2-fluorophenyl)-2-hydroxyethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
2-methyl-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-(thiophen-2-ylformamido)propanamide
(2R,3S,6R)-5-cyclobutanecarbonyl-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
7-(pyridin-3-yl)-4-(quinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
8-({3-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)quinoline
(2S)-2-amino-1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(1H-indol-3-yl)propan-1-one
2-({[(3R,4R)-4-(hydroxymethyl)-1-(3-methoxy-2-methylbenzoyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-({2-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine