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3-[(3S,4R)-4-(dimethylamino)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-1-[4-(2,5-dimethylphenyl)piperazin-1-yl]propan-1-one
3-{1-[3-(1H-imidazol-1-yl)propanoyl]piperidin-3-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({1-[2-(1H-1,3-benzodiazol-1-yl)acetyl]piperidin-3-yl}methyl)-4-methoxybenzene-1-sulfonamide
3-amino-N-({1-[(3,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)benzamide
1-(2-oxo-2-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethyl)-1,2-dihydropyrimidin-2-one
[2-(1-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidin-2-yl)ethyl]dimethylamine
(3aR,6aR)-2-(4-cyclobutyl-6-methylpyrimidin-2-yl)-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methyl-1-{[1-phenyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
dimethyl(3-{2-[1-(2-methylquinolin-4-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
(3S,4R)-3-ethyl-4-methyl-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-ol
(2S,4R)-N-ethyl-4-(3-methyloxetane-3-amido)-1-(2-phenylethyl)pyrrolidine-2-carboxamide
1-tert-butyl-4-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
4-[(4-fluorophenyl)methyl]-1-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-(3-fluorophenyl)piperidine
diethyl[1-(furan-2-yl)-2-(4H-1,2,4-triazol-4-yl)ethyl]amine
5-oxo-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
{2-[2-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}methanol
{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
4-(5-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}pyrimidin-2-yl)morpholine
6-chloro-8-methyl-3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,4-dihydroquinazolin-4-one
N-[(3R,4S)-4-cyclopropyl-1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)pyrrolidin-3-yl]-2-methoxyacetamide
4-benzyl-3-ethyl-1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]-1,4-diazepan-5-one
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
(3aR,5R,6S,7aS)-N-(5-acetamido-2-methoxyphenyl)-5,6-dihydroxy-octahydro-1H-isoindole-2-carboxamide
1-(cyclohexylmethyl)-3-hydroxy-3-({[2-(3-methylthiophen-2-yl)ethyl]amino}methyl)piperidin-2-one
6-methyl-2-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}pyridine-3-carboxylic acid
N-benzyl-N-methyl-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[3-(4-fluorophenyl)phenyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-3-carboxamide
N-{[7-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-methoxy-2-phenylacetamide
(3S)-1-(1-methyl-5-{6-oxa-9-azaspiro[4.5]decane-9-carbonyl}-1H-1,3-benzodiazol-2-yl)pyrrolidin-3-ol
{[7-chloro-2-(2-phenoxyethoxy)quinolin-3-yl]methyl}[3-(morpholin-4-yl)propyl]amine
(4aS,7aR)-4-ethyl-6,6-dioxo-N-[2-(propan-2-yl)phenyl]-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
5-ethyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
2-methyl-N-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]-2-(thiophen-2-ylformamido)propanamide
1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)ethan-1-one
{3-[(3-chlorophenyl)methyl]-1-(3,6-dimethylpyrazin-2-yl)piperidin-3-yl}methanol
9-methoxy-3-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-{4-[2-(pyridin-3-yl)-1H-imidazol-1-yl]butyl}azepane
4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-5-methyl-N-[(3-methylphenyl)methyl]thieno[2,3-d]pyrimidine-6-carboxamide
2-[3-(3-fluorophenoxymethyl)-5-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
6-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2H-1,3-benzodioxol-5-amine
4-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
1-(4-chloro-2-fluorobenzoyl)-3-(2-ethylphenoxy)azetidine
N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}furan-2-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
4-(4-{[2-(methoxymethyl)piperidin-1-yl]methyl}phenyl)-2-methylbutan-2-ol
1-benzyl-N3-cyclohexyl-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(1R,5R)-6-(2-methoxyethyl)-3-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-3,6-diazabicyclo[3.2.2]nonane