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4-(4-benzyl-1H-1,2,3-triazol-1-yl)-1-(oxan-4-yl)piperidine
N-[(3R,4S)-1-(4-aminopyrimidin-2-yl)-4-cyclopropylpyrrolidin-3-yl]cyclopropanesulfonamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-oxo-1,3-oxazolidine-4-carboxamide
1-methyl-4-(2-{1-[(3-methylphenyl)methyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}ethyl)piperazine
4-{[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
5-(4-{[1-(4-methoxyphenyl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
N-[4-({[2-(propan-2-yloxy)ethyl]carbamoyl}methoxy)phenyl]propanamide
methyl 3-(1-methylcyclohexanecarbonyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
9-(2-hydroxypropyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-5-({[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)furan-2-carboxamide
1-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)ethan-1-one
2-{[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]methyl}-6-methylpyridin-3-ol
3-(1-methyl-1H-imidazol-2-yl)-6-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}pyridazine
3-(2-methylphenyl)-3-phenyl-1-(pyrrolidin-1-yl)propan-1-one
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
7-(1-benzothiophen-3-yl)-4-cyclobutanecarbonyl-9-ethoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[1-(3-methylphenyl)-5-oxo-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-[2-(pyridin-2-yl)ethyl]acetamide
4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine
1-methyl-4-[(5-methylthiophen-2-yl)methyl]-2-phenylpiperazine
N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-4-[4-(trifluoromethyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 5-{4-[(3,4-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}-5-oxopentanoate
N-[(3S,4R)-1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-4-propylpyrrolidin-3-yl]methanesulfonamide
9-[3-(methylsulfanyl)propanoyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(3-chlorophenyl)-4-[2-(3-fluoro-4-hydroxyphenyl)acetyl]piperazin-2-one
N-methyl-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(1H-pyrazol-4-yl)ethyl]pyridin-2-amine
1-(2,2-diphenylethyl)-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
1-[5-(2-chlorophenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]butan-2-ol
5-fluoro-2-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
2,3,5-trimethyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}pyrazolo[1,5-a]pyrimidin-7-amine
(3S)-3-{[1-methyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}azepan-2-one
9-[(2S,4S)-4-amino-1-methylpyrrolidine-2-carbonyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(2R,3R,6R)-5-[(4-methyl-1H-imidazol-5-yl)methyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
2-(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carbonyl)pyridine
3-(2H-1,3-benzodioxol-5-yl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}propanamide
N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]cyclohexanecarboxamide
3-(3-methoxybenzoyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine
2-(4-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}morpholin-3-yl)acetic acid
4-(2,3-dihydro-1H-indene-1-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
4-cyclobutanecarbonyl-1-(2-methylphenyl)piperazin-2-one
4-[2-(4-phenylpiperidin-1-yl)ethyl]thiomorpholine
N4-[3-(propan-2-yloxy)propyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
4,6-dimethyl-2-[6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-2-yl]pyridine-3-carbonitrile
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
3-{1-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-3-yl}benzoic acid
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(6-methylpyridazin-3-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
{3-[(4-fluorophenyl)methyl]-1-(isoquinoline-1-carbonyl)piperidin-3-yl}methanol
[4-(2-phenylethyl)-1-[2-(1H-1,2,3,4-tetrazol-1-yl)pyridine-4-carbonyl]piperidin-4-yl]methanol
N-[2-(4-chlorophenyl)ethyl]-1-methylazepane-2-carboxamide