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4-(1H-imidazol-1-ylmethyl)-1-[(6-methoxypyridin-3-yl)methyl]piperidin-4-ol
4-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}thiomorpholine
N-{2-[({2-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)amino]ethyl}acetamide
1-methyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4,6-dimethyl-3-[(2S)-2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
6,7-dimethoxy-2-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-1,2,3,4-tetrahydroisoquinoline
4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
3-(2-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-oxoethyl)-1-cyclopropyl-3-(4-methoxyphenyl)pyrrolidine-2,5-dione
3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-methyl-1-[3-(1H-pyrazol-1-yl)phenyl]urea
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-[4-(propan-2-yl)-1,3-thiazol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
6-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
4-methoxy-N-{1-[1-(thiophene-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
(3R,4R)-1-(5-fluoro-2-methylbenzenesulfonyl)-3,4-dimethylpyrrolidin-3-ol
5-oxo-1-(pyridin-2-ylmethyl)-N-[3-(pyridin-3-yloxy)propyl]pyrrolidine-3-carboxamide
N,N,4-trimethyl-3-{[(1,2-oxazol-5-ylmethyl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}pyridin-2-amine
2-[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]-1-(pyridin-3-yl)ethan-1-ol
2-[1-(2-fluorophenyl)-5-(oxan-2-yl)-1H-1,2,4-triazol-3-yl]acetamide
[1-(5-methylpyrazine-2-carbonyl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
(3aS,6aS)-2-(1-propylpiperidin-4-yl)-5-(pyridin-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-fluoro-N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]quinoline-2-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-7-acetamido-N-methyl-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
N2,N2,N4-trimethyl-N4-[2-(methylsulfanyl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-(pyridin-3-yl)acetamide
N-[4-(1H-1,2,4-triazol-1-yl)phenyl]morpholine-2-carboxamide
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
9-methoxy-3-[(4-methoxyphenyl)methyl]-7-oxo-N-[3-(1H-pyrazol-1-yl)propyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-methyl-1H-1,3-benzodiazole
{1-[(4-ethylphenyl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
(2E)-1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-phenylprop-2-en-1-one
1-{[2-(difluoromethoxy)phenyl]methyl}-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N-(3-{4-[(2-methoxy-2-phenylacetamido)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)-3-(pyridin-3-yl)propanamide
[(1-benzyl-1H-imidazol-2-yl)methyl](1H-imidazol-4-ylmethyl)methylamine
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]butanamide
6-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
1-[6-methyl-3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)quinolin-2-yl]piperidin-3-ol
2-{[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetic acid
3-[2-(dimethylamino)ethyl]-1-ethyl-8-(furan-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperazin-1-yl}-1-azabicyclo[2.2.2]octane
1-ethyl-5-[2-(2H-indazol-2-yl)acetyl]-N-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-methyl-4-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-1,4,9-triazaspiro[5.5]undecane
(2S)-1-[4-(4-ethoxy-3-methylphenyl)-4-oxobutanoyl]pyrrolidine-2-carboxylic acid
N-(2-methoxyethyl)-3-({1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}oxy)benzamide
[(3-methoxyphenyl)methyl](methyl){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
5-methyl-3-{[2-(6-methylhept-5-en-2-yl)-1H-imidazol-1-yl]methyl}-1,2-oxazole
(1S,5R)-6-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(cyclohexylmethyl)-N-(9H-fluoren-9-yl)-1H-1,2,3-triazole-4-carboxamide
(2S)-1-{2-[N-(4-methylphenyl)methanesulfonamido]acetyl}pyrrolidine-2-carboxamide
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2,3-dimethyl-1H-indole-5-carboxamide