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2-[(4-benzylpiperazin-1-yl)methyl]-N-cycloheptyl-1,3-oxazole-4-carboxamide
N-(3-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-3-oxopropyl)-N-methylmethanesulfonamide
6-(1H-indazol-5-yl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-hydroxy-1-(quinoxalin-2-yl)piperidine-4-carboxylic acid
7-(cyclopropylmethyl)-2-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetyl)-2,7-diazaspiro[4.5]decan-6-one
4-(azepan-1-yl)-7-(furan-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
2-{4-[3-(furan-2-yl)propyl]piperazin-1-yl}pyrimidine
(2S)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
5-[(dimethylamino)methyl]-N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)furan-2-carboxamide
N-[(3R,5S)-1-[(2E)-but-2-en-1-yl]-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
ethyl 5-[({5-[(2-methylpropyl)carbamoyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridin-3-yl}formamido)methyl]furan-2-carboxylate
4-{[(5-fluoropyridin-3-yl)carbamoyl]amino}-N-methylbutanamide
2-(dimethylamino)-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-2-(2-methylphenyl)acetamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-3-yl]methanol
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(2-methoxyphenoxy)ethan-1-one
4-hydroxy-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)pyrimidine-5-carboxamide
N-(butan-2-yl)-5-(morpholin-4-ylmethyl)-N-(pyridin-3-ylmethyl)furan-3-carboxamide
N-(prop-2-en-1-yl)-2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}aniline
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,4-dimethylphenyl)urea
N-[(2,6-dimethoxyphenyl)methyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
3-{4-[1-(oxan-4-yl)piperidine-3-carbonyl]piperazin-1-yl}phenol
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-(2-methoxyphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-(2-methoxyphenyl)-N-(pyridin-3-ylmethyl)acetamide
(2R)-1-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetyl]pyrrolidine-2-carboxamide
3-methyl-4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-{3,9-diazaspiro[5.5]undecan-3-yl}-3-(morpholin-4-yl)propan-1-one
4-methyl-1-(2-{1-oxa-8-azaspiro[4.5]decan-8-yl}-2-oxoethyl)-1,2-dihydroquinolin-2-one
4-{5-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
N-[(3,5-dimethoxyphenyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-3-carboxamide
3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]urea
2-[(cyclopentylamino)methyl]-4-(pyridin-2-yl)phenol
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]methanol
3-[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]pyridine
3-({1-[(2-aminopyridin-3-yl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
1-(4-chlorophenyl)-N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopropane-1-carboxamide
2-{[1-(pyrazin-2-yl)propan-2-yl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(2S,4R)-4-amino-N-ethyl-1-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)pyrrolidine-2-carboxamide
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
3-{4-[5-(3-fluorobenzamido)-1H-pyrazol-1-yl]piperidin-1-yl}propanoic acid
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(3,4-dimethoxyphenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
1-[(3,4-difluorophenyl)methyl]-3-[4-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
4-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]-N-cyclohexylpiperidine-1-carboxamide
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-2-[3-(trifluoromethyl)phenyl]acetamide
2-(4-fluorophenyl)-N,N-dimethylpiperidine-1-carboxamide
1-[(2-chlorophenyl)methyl]-N-methyl-N-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-N-{2-[(4-methylphenyl)sulfanyl]ethyl}pyrimidin-2-amine
1-[3-(pyridin-3-yl)propyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one