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N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2-methyl-N-(2-methylpropyl)-1H-pyrrole-3-carboxamide
methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}amine
3-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-1,2-benzoxazole
2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]ethan-1-one
6-{[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]methyl}-2-oxo-N-[(1r,4r)-4-hydroxycyclohexyl]-1,2-dihydropyridine-3-carboxamide
2-[(3,3-dimethyl-3,4-dihydroisoquinolin-1-yl)methyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(1,3-oxazole-5-carbonyl)piperidine
N-(1,4-dimethyl-1H-pyrazol-5-yl)-2-{3-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}acetamide
5-fluoro-2-{[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}-3-methyl-1H-indole
N-ethyl-1-[3-(furan-2-yl)phenyl]-N-methylpiperidin-4-amine
(4aS,8aR)-1-(3-aminopropyl)-6-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-decahydro-1,6-naphthyridin-2-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[3-(dimethylamino)benzoyl]pyrrolidin-3-yl]methanol
3-[(1S,3S,3aR,6aS)-3-(hydroxymethyl)-5-methyl-3-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]phenol
2-(2,4-dimethoxyphenyl)-1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]ethan-1-one
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-methoxy-N,N-dimethyl-5-({[2-(pyridin-3-yloxy)propyl]carbamoyl}amino)benzamide
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(pyrrolidine-1-carbonyl)piperidine-4-carboxylic acid
N-[(2R,3R)-1'-[2-(2-fluorophenyl)acetyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxyacetamide
5-fluoro-2-{2-[(6-methoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]phenyl}-6-methyl-3,4-dihydropyrimidin-4-one
1-cyclopentyl-3-(3-methoxyphenyl)-3-[2-oxo-2-(3-oxo-4-phenylpiperazin-1-yl)ethyl]pyrrolidine-2,5-dione
2-phenoxy-N-(2-{7-[(2,3,4-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
4-[3-cyclopropyl-5-(3-phenyl-1H-pyrazol-4-yl)-1H-1,2,4-triazol-1-yl]-3-methylpyridine
3-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-2H-indazole
N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-1-(pyrimidin-2-yl)piperidin-4-amine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methyl-2-(trifluoromethyl)pyrimidin-4-amine
ethyl 3-[(2-methylphenyl)methyl]-1-(thiophene-2-sulfonyl)piperidine-3-carboxylate
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-4-(naphthalen-1-yl)-4-oxobutanamide
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-N-(pyridin-2-ylmethyl)acetamide
6-methyl-4-[3-(pyrimidin-4-yl)piperidin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
N-cyclooctyl-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-chlorobenzamide
(4aS,8aR)-1-(3-aminopropyl)-6-(3-phenyl-1,2,4-oxadiazol-5-yl)-decahydro-1,6-naphthyridin-2-one
(4aS,7aR)-1-[(2,6-dimethoxyphenyl)methyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperazine-2-carboxylic acid
4-(6-methylpyridine-2-carbonyl)-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
1-{[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenyl]methyl}piperidine
5-cyclohexaneamido-N-[2-(furan-2-yl)ethyl]-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
N-methyl-1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-N-(2-phenylethyl)piperidin-3-amine
3-{2-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]ethyl}quinoxalin-2-ol
4-({2-[2-(4-chlorophenyl)pyrimidin-5-yl]-1H-imidazol-1-yl}methyl)-1-methylpiperidin-4-ol
3-{1-[1-(1-benzofuran-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
3,6,7-trimethyl-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1-benzofuran-2-carboxamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2-(1H-imidazol-2-yl)benzamide
3-{2-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-3,4,5-trimethoxybenzamide
N-{[7-chloro-5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylfuran-2-carboxamide
5-cyclopropanecarbonyl-1'-[(2-fluoro-4-methoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
5-(1-benzyl-1H-pyrazole-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid