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N-(1-{2-[3-(2-chlorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-3-(2-methoxyphenyl)propanamide
N-[(2R,3R)-1'-(1H-indole-2-carbonyl)-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
3-(1,4-diazepane-1-sulfonyl)-N-(2,2,2-trifluoroethyl)benzamide
{1-[({[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]cyclopropyl}methanol
{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-2-phenylethyl}(methyl)(pyridin-4-ylmethyl)amine
3-[1-(4-methylpyridin-2-yl)-1H-imidazol-2-yl]benzoic acid
N,N-dimethyl-5-{[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]methyl}pyrimidin-2-amine
ethyl 1-(2,5-dimethylfuran-3-carbonyl)-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
(1S,5R)-6-benzyl-3-(1-methyl-1H-indole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-4-yl)-N-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]acetamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-(furan-2-ylmethyl)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-chloro-N-ethyl-5-({[3-(1H-imidazol-2-yl)propyl]carbamoyl}amino)benzamide
3,5-dimethyl-2-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]-1H-indole
1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N-(isoquinolin-5-ylmethyl)-N-methyl-3-propyl-1H-pyrazole-4-carboxamide
N-[(2-fluorophenyl)methyl]-1-(6-methoxy-4-methylquinazolin-2-yl)piperidin-4-amine
ethyl 1-[3-(2-oxopiperidin-1-yl)propanoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
5-methyl-1-{2-oxo-2-[2-(3-phenylpropyl)morpholin-4-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-2-(2,3,6-trimethylphenoxy)acetamide
3-(oxan-4-yl)-5-[4-(1H-pyrazol-1-yl)phenyl]-1H-1,2,4-triazole
(2,1,3-benzothiadiazol-5-ylmethyl)({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
2-{[({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-4-methoxyphenol
methyl 4-{[methyl({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}-1H-pyrazole-3-carboxylate
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-3-(1,2-oxazolidin-2-yl)propanamide
3-[4-(1,2-benzothiazol-3-yl)piperazine-1-carbonyl]piperidine-1-carboxamide
1-{1-[(2-methylnaphthalen-1-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
(1S,5R)-3-(5-acetyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,3S)-2-amino-1-[4-({4-[(dimethylamino)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidin-1-yl]-3-methylpentan-1-one
7-methyl-2-[2-(2-oxo-1,2,3,4-tetrahydroquinolin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-({1-[3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanoyl]piperidin-3-yl}methyl)-1H-indole-2-carboxamide
14-(4-fluoro-3-methylphenyl)-5-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
5-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
5-methyl-4-(5-methyl-1,3-oxazole-4-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
(3aR,6aR)-2-(2-hydroxyethyl)-5-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-ethoxy-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
3-[3-(pyridin-2-yl)phenyl]-1-[(1r,4r)-4-hydroxycyclohexyl]urea
2-({2-[4-(2-ethylpyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}amino)-6-methyl-3,4-dihydropyrimidin-4-one
2-phenyl-4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]morpholine
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3,5-difluoropyridine-2-carboxamide
1-methyl-N-[(4-methyl-1H-imidazol-5-yl)methyl]-N-(pyridin-3-ylmethyl)piperidin-4-amine
4-[(4-methyl-5-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
N-ethyl-2-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(thiophen-2-ylformamido)propanamide
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)pyridine-3-carboxamide
3-(cyclopropylmethyl)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidine-3-carboxylic acid
2-(1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethan-1-ol
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
3-{1-[(2-chloro-4-hydroxy-5-methoxyphenyl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
4-[2-methyl-2-(piperidin-1-yl)propyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
9-(5-ethyl-2-methylpyrimidin-4-yl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2-{1-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide