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2-[2-(pyridin-4-yl)ethyl]-9-(thiophene-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(1H-imidazol-1-yl)propyl]-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
2-(2-hydroxyacetyl)-N-methyl-N-(pyridin-3-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-methyl-N-(quinolin-5-ylmethyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
4-[(4-methyl-1H-pyrazol-1-yl)methyl]-N-(4-oxo-4H-chromen-6-yl)piperidine-1-carboxamide
methyl 3-(2-methoxyacetamido)-1-methyl-5-[(5-methylhex-5-en-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{1'-[2-(ethylamino)pyrimidine-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
(4aR,7aS)-1-(2-methoxyacetyl)-4-(thiophen-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(2,2-diphenylacetyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(6-chloropyridin-3-yl)-3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
2-ethoxy-3-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]pyridine
1-({1-methyl-4-oxo-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-6-yl}methyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(1R,5R)-6-[3-(3-fluorophenyl)propanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-{[2-(4-fluorophenyl)pyrrolidin-1-yl]sulfonyl}-4-methoxypiperidine
4-(1-{4-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]phenyl}ethyl)morpholine
5-(1-{[4-(diethylamino)phenyl]methyl}piperidin-4-yl)-5-(3-phenylpropyl)imidazolidine-2,4-dione
(1S,5R)-3-(2-methylbenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[(4aR,8aR)-7-(4-aminopyrimidin-2-yl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]acetic acid
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
7-(2-methylphenyl)-4-[6-(propan-2-yl)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[1-(2-chlorophenyl)ethyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}acetamide
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
5-methyl-3-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,2-oxazole
3-chloro-6-{4-[(5-ethylpyridin-2-yl)methyl]piperazin-1-yl}pyridazine
N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-cyclopropylmethanesulfonamide
2-phenoxy-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
(4aR,8aR)-2-methanesulfonyl-7-[2-(6-methylpyridin-2-yl)ethyl]-decahydro-2,7-naphthyridin-4a-ol
4-fluoro-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-methoxy-N-methylbenzamide
N-[cyclopropyl(4-methoxyphenyl)methyl]-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
(2S,4R)-N-methyl-1-(2-methylpropyl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(2R,3R)-3-(1,2,3,6-tetrahydropyridin-1-yl)-1'-(thiophen-2-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-fluoro-N-[(2R,3R)-2-methoxy-1'-[(2E)-2-methylbut-2-en-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
(3S,4S)-4-{[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}-1-[(5-propylfuran-2-yl)methyl]pyrrolidin-3-ol
N,1,6-trimethyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-4-(thiophen-2-yl)butan-1-one
2-methyl-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1H-1,3-benzodiazole
1,3-dimethyl-N-[2-(3-methylpyridin-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)(methyl)[(3,4,5-trimethoxyphenyl)methyl]amine
N-(4-{[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]methyl}phenyl)acetamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-(2-hydroxy-3-methoxypropyl)benzamide
2-(dimethyl-1,2-oxazol-4-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
1-cyclopentyl-4-[2-(1H-1,2,4-triazol-5-yl)benzoyl]piperazin-2-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-[3-(2-fluorophenyl)propanoyl]piperidin-3-yl]propanoic acid
N-benzyl-N-butyl-2-[3-(3-fluorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]acetamide
(3aS,6aR)-3-cyclopentyl-5-(3,6-dimethylpyrazin-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-(cyclopropylmethyl)-5-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-1-(propan-2-yl)-1H-1,2,4-triazole
6-(2-aminoethyl)-N,2-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyrimidin-4-amine