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5-hydroxy-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyridine-2-carboxamide
1-methyl-N-[(5-methylpyrazin-2-yl)methyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-(1-methylpyrrolidin-2-yl)acetamide
5-(2-methylfuran-3-carbonyl)-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)naphthalene-1-carboxamide
7-(5-chloropyridin-2-yl)-4-(2-phenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4-methylpiperidine-4-carboxamide
3-(1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-[2-(2-methoxyquinolin-3-yl)-1H-imidazol-1-yl]-N,N-dimethylethane-1-sulfonamide
methyl 7-oxo-3-[2-(pyrimidin-2-ylsulfanyl)acetyl]-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
7-(cyclopropylmethyl)-2-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)-2,7-diazaspiro[4.5]decan-6-one
1-[3-(2-oxopyrrolidin-1-yl)propyl]-5-[4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carbonyl]piperidin-2-one
3-{1-[1-(3-cyclopentylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
2-({3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)pyridine-3-carboxylic acid
1-[(2-methoxyphenyl)methyl]-N3-(3-methylbutyl)-4-oxo-N5-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)pent-4-enamide
methyl 7-oxo-3-(1,3-thiazole-4-carbonyl)-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-N-ethyl-4-methyl-1,3-thiazol-2-amine
3-phenyl-N-[4-(4-{[3-(pyridin-3-yloxy)propyl]amino}piperidin-1-yl)phenyl]propanamide
(2E)-1-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-3-(pyridin-4-yl)prop-2-en-1-one
3-(4-fluorophenyl)-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-phenylpropanamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
2-{2-chloro-4-[(4-phenyl-1,4-diazepan-1-yl)methyl]phenoxy}acetamide
3-benzoyl-1-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]piperidine
N-[2-(4-ethylmorpholin-2-yl)ethyl]-2-(methylamino)pyridine-3-carboxamide
N-[(5-methylpyrazin-2-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
2-[1-(2-chlorophenyl)-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
N-[3-(methylsulfanyl)propyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
4-[4-(benzenesulfonyl)piperazin-1-yl]-5-ethyl-2-methylpyrimidine
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-[1-(4-methylbenzoyl)piperidin-4-yl]imidazolidine-2,4-dione
4-(cyclopropylmethyl)-1-(4-methoxypyrimidin-2-yl)-3-(propan-2-yl)-1,4-diazepan-5-one
4-sulfamoyl-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
N-(1,3-benzothiazol-2-ylmethyl)-3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{1-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
1-(4-methoxy-3,5-dimethylbenzoyl)-N,N-dimethylazepan-4-amine
2-phenyl-N-[3-(1H-pyrazol-1-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3aS,6aS)-2-methyl-5-[2-(naphthalen-1-yl)ethanesulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[1-(propan-2-yl)piperidine-4-carbonyl]piperidine
2-(1H-indol-3-yl)-1-(4-{2-[(2-methylphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)ethan-1-one
1-ethyl-3-(3-fluoro-4-methylphenyl)-6-[3-(methylsulfanyl)propyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
3-[5-oxo-2-(thiophen-3-ylmethyl)pyrrolidin-2-yl]-N-{2-[4-(trifluoromethyl)phenyl]ethyl}propanamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
3-methyl-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
N-{[3-methyl-7-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-carboxamide
4-[(4-fluorophenyl)methyl]-1-[2-(1H-imidazol-1-yl)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-{2-[(5-ethylpyrimidin-2-yl)amino]ethyl}piperidin-4-ol
2-(ethoxymethyl)-N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-methyl-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-3-phenylpiperidine