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3-methyl-3-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1-[4-(2-methylpropoxy)phenyl]urea
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
7-fluoro-3-(morpholin-4-ylmethyl)-1-(pyridin-4-ylmethyl)-1,2-dihydroquinolin-2-one
2-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]-4,5,6,7-tetrahydro-1,3-benzothiazole
7-(1,3-benzothiazol-2-yl)-4-[1-(4-chlorophenyl)cyclopropanecarbonyl]-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3aR,6aR)-2-[(dimethyl-1,3-thiazol-4-yl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-({7-[(4-fluoro-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-(3-fluorophenyl)acetamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-(2-oxoimidazolidin-1-yl)benzamide
1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one
N-[(3R,4S)-4-cyclopropyl-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl]pyrazine-2-carboxamide
5-{5-[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
methyl 3-[2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamido]propanoate
1-(4-benzylpiperazin-1-yl)-3-[1-(furan-3-ylmethyl)piperidin-3-yl]propan-1-one
1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-4-(pyrrolidin-1-yl)pentan-1-one
1-benzyl-3-methyl-8-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(4-{2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]acetyl}piperazin-1-yl)propanamide
1-{3,5-dimethyl-4-[2-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1H-pyrrol-2-yl}ethan-1-one
(4aR,7aS)-1-ethyl-4-(3-{[(4-fluorophenyl)methyl]sulfanyl}propanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-cyano-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)-N-cyclohexylpropanamide
3-[5-oxo-2-(thiophen-3-ylmethyl)pyrrolidin-2-yl]-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
N-[2-(methylamino)ethyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
3-{1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-(2-methoxyphenyl)-3-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}formamido)propanamide
(2E)-1-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)prop-2-en-1-one
1-[(4aS,8aS)-4a-hydroxy-7-[(1-methyl-1H-imidazol-2-yl)methyl]-decahydro-2,7-naphthyridin-2-yl]-2-(methylsulfanyl)ethan-1-one
N-methyl-N-({2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl}methyl)oxan-4-amine
4-cyano-N-(3-methoxy-4-methylphenyl)piperidine-1-carboxamide
N-[2-(dimethylamino)ethyl]-4-{[(3R)-pyrrolidin-3-yl]sulfamoyl}benzamide
methyl 2-({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amino)pyridine-4-carboxylate
2-{3-[4-(benzyloxy)piperidine-1-carbonyl]piperidin-1-yl}-4,7-dimethylquinazoline
2-[4-(2-{[(2-chlorophenyl)methyl]sulfanyl}acetyl)morpholin-3-yl]acetic acid
4-{5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(2-methoxyacetyl)-2,8-diazaspiro[4.5]decan-3-one
2-[(4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}phenyl)formamido]-N,N-dimethylacetamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-amine
1-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-4-(pyridin-4-yl)piperazine
(1S,5R)-N,N-dimethyl-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-sulfonamide
N-{1-[1-(quinolin-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}pyridine-3-carboxamide
1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-2-ethylpiperidine
(3S,4R)-1-(2,6-dimethoxypyridine-3-carbonyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
N-[(1-ethyl-1H-indazol-3-yl)methyl]-2-(methylamino)pyridine-4-carboxamide
N,6-dimethyl-2-oxo-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
5-phenyl-N-[4-(4-{[2-(pyridin-3-yloxy)ethyl]amino}piperidin-1-yl)phenyl]pentanamide
3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(4-methoxyphenyl)ethyl]-1-methyl-N-[(1-methylpiperidin-4-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-[3-(methylsulfanyl)propyl]acetamide
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-[4-(dimethylamino)phenyl]-1-(1-methylpiperidin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
9-(cyclopropanesulfonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
6,7-dimethyl-2-{[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]methyl}-1H-1,3-benzodiazole