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N-(3,3-diphenylpropyl)-2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-6-methylphenol
3-(3-methoxyphenyl)-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1H-pyrazole-5-carboxamide
6-(methoxymethyl)-1-methyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
5-chloro-3-[1-(6-methylpyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
1-[(2-fluoro-5-methoxyphenyl)methyl]-4-(2-methylpropyl)-1,4-diazepan-5-one
2-{5-[2-(2-methylphenyl)phenyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-{4-[(2,4-dimethoxyphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
1-[2-chloro-5-(trifluoromethyl)benzoyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
2-(propan-2-yloxy)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}ethan-1-one
1-[(2-fluorophenyl)methyl]-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
1-benzyl-8-(propan-2-yl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-hydroxyethyl)-9-[3-(4-hydroxyphenyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2-fluoro-5-methylphenyl)-3-(piperidin-1-yl)pyrrolidine-1-carboxamide
N-(1-{7-[(2-hydroxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
ethyl 1-(5-ethanesulfonamido-1-methyl-2-phenyl-1H-1,3-benzodiazole-7-carbonyl)piperidine-3-carboxylate
4-(pyrrolidin-1-yl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
(3S,4R)-4-(2-methylphenyl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}pyrrolidine-3-carboxylic acid
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
3-(3-chlorobenzoyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
3-[2-(adamantan-1-yl)acetamido]butanoic acid
8-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
(2R,3R,6R)-N,N-dimethyl-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
3-(hydroxymethyl)-3-methyl-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
N-(oxolan-2-ylmethyl)-1-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)piperidine-4-carboxamide
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]acetamide
5-ethyl-2,4-dimethyl-6-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}pyrimidine
2-methyl-N-(pyridin-4-ylmethyl)-1-benzofuran-7-carboxamide
5-[4-hydroxy-1-(2-phenylpropyl)piperidin-4-yl]-N-(pyridin-4-ylmethyl)-1-benzofuran-2-carboxamide
6-(cyclopent-1-ene-1-carbonyl)-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
2-(adamantan-1-yl)-4-hydroxy-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]pyrimidine-5-carboxamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-methyl-4-{[(4-phenylphenyl)methyl]amino}pyrrolidine-2-carboxamide
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[(3-methyl-1,2-oxazol-5-yl)methyl]amine
2-cyclopentyl-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)acetamide
1-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-N-(propan-2-yl)-1H-pyrrole-2-carboxamide
2-(2,4-dimethoxyphenyl)benzonitrile
N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-{4-[({1-[(4-chlorophenyl)methyl]piperidin-3-yl}amino)methyl]phenoxy}ethan-1-ol
2-[5-(1-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
5-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole
3-(2-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)pyridine
ethyl 2-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}morpholin-3-yl)acetate
(1R,7S)-6-(azetidine-1-carbonyl)-3-[2-(pyridin-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-(2,1,3-benzoxadiazole-4-sulfonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-({8-[(3,5-dimethylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)oxolane-2-carboxamide
methyl (2S,4R)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-{2-[4-(trifluoromethyl)phenyl]benzamido}pyrrolidine-2-carboxylate
2-{2-[4-phenyl-1-(pyrrolidin-3-yl)-1H-imidazol-5-yl]-1H-pyrrol-1-yl}-1,3-thiazole
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}acetamide
3-(1-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-1H-1,2,3-triazol-4-yl)piperidine