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(1S,5R)-6-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
1-methyl-4-(1,3,7-trimethyl-1H-indole-2-carbonyl)-1,4,9-triazaspiro[5.5]undecane
N'-(3-chloro-4-fluorophenyl)-N-[1-(1H-pyrazol-1-yl)propan-2-yl]butanediamide
3-[1-(furan-3-carbonyl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
1-[(2-chlorophenyl)methyl]-N-[2-(4-hydroxypiperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(6-methoxypyridin-3-yl)-7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
1-(adamantan-2-yl)-4-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
N,N,4-trimethyl-5-[4-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]pyrimidin-2-amine
2-{1-[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
1-(prop-2-en-1-yl)-N-[3-(pyrrolidin-1-yl)propyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4aS,7aR)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}({2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl})amine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
1-[(1R,3R,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-2-(morpholin-4-yl)ethan-1-one
N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
2-methyl-3-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-2,8-diazaspiro[4.5]decane
3-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-2-methylphenol
1-{1-[(3-methylpyridin-2-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
(4aR,7aS)-1-(2-hydroxyethyl)-4-(1-methyl-1H-indole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-6-(cyclopropylmethyl)-3-(2,5-dimethoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-methyl-6-(3-methylpiperazin-1-yl)-2-phenylpyrimidine
N-methyl-1-(naphthalen-1-ylmethyl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-{[1-(2-methoxyphenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]methyl}-6-methyl-2,3-dihydropyridazin-3-one
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
[4-({methyl[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)oxan-4-yl]methanol
5-chloro-6-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-2-methylpyrimidin-4-ol
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-methyl-N-[2-(4-methylphenoxy)ethyl]acetamide
2-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline
1-[2-(1,4-dioxo-1,2,3,4-tetrahydrophthalazin-2-yl)ethyl]-5-oxopyrrolidine-3-carboxylic acid
2-(4-fluorophenoxy)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
({5-[1-(3-chloropyridin-2-yl)piperidin-4-yl]-4-cyclopropyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
(4aR,7aS)-1-acetyl-4-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2-{[(4-cyano-2-ethylphenyl)carbamoyl]amino}ethyl)piperidine-3-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-methyl-1,3-benzoxazole-6-carboxamide
(1R,5R)-6-(2-ethylpyridine-4-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
methyl 9-[2-(2-fluorophenyl)ethoxy]-3-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-{[(5-ethylpyridin-2-yl)methyl](methyl)amino}-N-(1,3-thiazol-2-yl)propanamide
N-(1-hydroxybutan-2-yl)-8-oxo-7-(prop-2-en-1-yl)-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine
N-[4-(furan-2-yl)phenyl]-1-(1,2-oxazol-3-ylmethyl)piperidine-3-carboxamide
methyl (2S)-1-{[4-(2-ethylbutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}pyrrolidine-2-carboxylate
7-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-{3-[3-(2-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[1-(pyridin-2-yl)propan-2-yl]benzamide
[(1S,3S,3aS,6aR)-3-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
N-[(5-chloro-2,3-dimethoxyphenyl)methyl]-1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-{[8-(6-cyclopropylpyrimidin-4-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
1-[3-(3-methoxyphenyl)phenyl]-N-(oxan-4-yl)piperidin-4-amine