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{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-tert-butyl-5-oxopyrrolidine-3-carboxamide
N-[(3S,4R)-1-{[4-(2-aminoethyl)phenyl]methyl}-4-propylpyrrolidin-3-yl]acetamide
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-[5-benzyl-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-methyl-1,4-diazepane
4-(azepan-1-yl)-2-{[3-(methoxymethyl)piperidin-1-yl]methyl}quinazoline
1-[(3-methyl-1H-pyrazol-5-yl)methyl]spiro[azepane-4,2'-chromene]
2-methyl-N-[3-(N-methylacetamido)phenyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-[3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,5,6-trimethyl-1,2-dihydropyridin-2-one
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-[1-(methylsulfanyl)propan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(propan-2-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
6-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyrimidine-2,4-diamine
2-(3-fluoropyridin-4-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
4-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,2-dihydrophthalazin-1-one
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-4-(piperidin-1-ylmethyl)benzamide
1-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-3-[1-(pyridin-2-ylmethyl)piperidin-4-yl]urea
5-methyl-2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
4-methoxy-N-[2-(7-{[4-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
1-[(4-methyl-1H-imidazol-2-yl)methyl]-5,5-diphenylpiperidin-2-one
methyl 9-[2-(2-fluorophenyl)ethoxy]-3-(1H-indol-2-ylmethyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-1,2-oxazole-3-carboxamide
3-({[(2-fluorophenyl)methyl](2-methoxyethyl)amino}methyl)-N-methylpyridin-2-amine
5-methyl-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-1-propyl-1H-pyrazole-4-carboxamide
3-(2-fluorophenyl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-3-phenylpropanamide
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-4-oxo-N-(propan-2-yl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-(pyridin-2-ylmethyl)-1,4-diazepane
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-(1H-pyrazol-3-ylmethyl)benzamide
N-[3-(1H-indazol-1-yl)propyl]-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
N-cyclopropyl-1-{1-[(3-fluoro-5-methylphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-benzyl-N-methyl-3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]propanamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1r,4r)-4-[(heptan-4-yl)amino]cyclohexan-1-ol
1-[1-(2-methoxypyridine-4-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
4-[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-6-(4-methyl-1H-pyrazol-1-yl)pyrimidine
3-(1-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}piperidin-3-yl)-1-(morpholin-4-yl)propan-1-one
methyl(2-phenylethyl){[3-(thiomorpholine-4-carbonyl)-1,2-oxazol-5-yl]methyl}amine
1-{3-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-oxopropyl}azepan-2-one
3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}urea
1-cyclopentyl-N-methyl-N-(oxan-4-yl)-6-oxopiperidine-3-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-[1-(3-methylbutyl)piperidin-4-yl]imidazolidine-2,4-dione
N-(furan-2-ylmethyl)-5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-(prop-2-yn-1-yl)-1,2-oxazole-3-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
2-{[4-(2,6-diaminopyrimidin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
1-(2-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-[1-(2-phenylethyl)piperidin-3-yl]-4-(pyrrolidine-1-carbonyl)pyridin-2-amine
3-(4-methoxy-2-methylphenyl)-1-[(1-propyl-1,2,5,6-tetrahydropyridin-3-yl)methyl]urea
(1R,7S)-3-[(2,5-dimethylphenyl)methyl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidine-1-carbonyl]benzonitrile
(4S)-3,3,4-trimethyl-1-{[2-(morpholin-4-yl)quinolin-3-yl]methyl}piperidin-4-ol
N-benzyl-2-[4-(4-{[2-(pyridin-3-yloxy)ethyl]amino}piperidin-1-yl)phenyl]acetamide