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1-(2-chlorophenyl)-4-[(2-fluoro-4,5-dimethoxyphenyl)methyl]piperazin-2-one
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
N-[(2-ethoxypyridin-3-yl)methyl]-6-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[2-hydroxy-2-(4-methoxyphenyl)propyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-{4-[(1,4-dithiepan-6-yl)amino]piperidin-1-yl}pyridine-3-carbonitrile
3-{1-butyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}pyridine
3-[1-(2-methylpropyl)-1H-pyrazol-5-yl]-1-(oxolan-2-ylmethyl)-1-[(2E)-3-phenylprop-2-en-1-yl]urea
N,N,4-trimethyl-5-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]pyrimidin-2-amine
N-(cyclohexylmethyl)-1-[2-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-4-carboxamide
({5-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-4-yl]-4-ethyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-[(5-ethylpyridin-2-yl)methyl]-N-[(2-methoxyphenyl)methyl]cyclopropanamine
6-{[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}naphthalen-2-ol
ethyl 2-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]amino}acetate
4-{1-[2-(2-hydroxyethoxy)ethyl]-4-phenyl-1H-imidazol-5-yl}-2-methoxy-6-(prop-2-en-1-yl)phenol
N-benzyl-N-(2-hydroxyethyl)-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-ethyl-4-hydroxy-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
3-[2-(dimethylamino)ethyl]-1-(3-methylbutyl)-8-[(3,4,5-trimethoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(but-2-yn-1-yl)-5-{1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}-5-[(3-fluorophenyl)methyl]imidazolidine-2,4-dione
3-[4-(1-ethyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]-1-azabicyclo[2.2.2]octane
4-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}thiomorpholine
4-benzyl-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-ethyl-5-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
3-(2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-5-methyl-2,3-dihydro-1H-indol-2-one
methyl 3-[(2,4-difluorophenyl)methyl]-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-N-[1-(1,3-thiazol-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
ethyl 5-{[(1-cyclopentyl-6-oxopiperidin-3-yl)formamido]methyl}furan-2-carboxylate
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-[4-(propan-2-yl)-1,3-thiazol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-ethyl-N-(pyridin-4-ylmethyl)-5-({[3-(trifluoromethyl)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]propanamide
(5S,9aS,9bS)-5-(1-benzofuran-2-yl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{[3-methyl-7-(3-phenylpropanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
5-[({[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
2-[2-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-6-methoxyphenoxy]propanoic acid
N-(2-methanesulfonylethyl)-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(1,2-benzoxazol-3-yl)-N-[1-(pyridin-2-yl)propan-2-yl]acetamide
N-butyl-3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
N-[(3R,4S)-1-(6-aminopyrimidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-(piperidin-1-yl)acetamide
3-{5-[(2-aminopyridin-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-cyclopropylpropanamide
3-[3-(dimethylamino)propyl]-8-(oxan-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[1-(4-fluorobenzoyl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
5-{4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-[3-(1H-indazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[(2R,3R,6R)-5-[(4-methyl-1H-imidazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
2-{3-[2-(2-fluoro-4,5-dimethoxyphenyl)-1H-imidazol-1-yl]phenyl}-N-methylacetamide
1-{3-[(4-fluorophenyl)methyl]-1,2-oxazole-5-carbonyl}-3-phenylpiperidine
4-(2,6-dimethoxybenzoyl)-9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-ethyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-1H-pyrazole-3-carboxamide
N-methyl-1-propyl-N-[1-(thiophen-2-yl)ethyl]-1H-pyrazole-5-carboxamide