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N,N,8-trimethyl-2-[1-(2-methylpyridin-4-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({[4-(1H-pyrazol-1-yl)phenyl]methyl})amine
(1-methyl-1H-imidazol-2-yl)(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidin-4-yl)methanol
3-phenyl-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
ethyl 2-(4-{1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidine-4-carbonyl}morpholin-3-yl)acetate
3-(3-{[3-(dimethylamino)propyl](methyl)amino}piperidine-1-carbonyl)-N-methylpyridin-2-amine
6-(2,3-dimethoxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
9-(3-chloro-4-methoxybenzoyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
2-(3-methyl-1,2-oxazol-5-yl)-1-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]ethan-1-one
2-(3-methoxypropyl)-9-[(3-methylpyridin-4-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(2-methylphenyl)ethyl]-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
5-{1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperidin-4-yl}-5-[(2-chlorophenyl)methyl]imidazolidine-2,4-dione
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-cyclopropylacetamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-6-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
5-(furan-2-ylmethyl)-5-[3-oxo-3-(4-phenylpiperidin-1-yl)propyl]pyrrolidin-2-one
N-{3-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-oxopropyl}methanesulfonamide
4-{5-[(4-benzylpiperidin-1-yl)methyl]-1,2-oxazole-3-carbonyl}-1,3-dimethylpiperazin-2-one
3-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]-2,1,3-benzothiadiazole-4-sulfonamide
N-[(2R,3R)-2-methoxy-1'-[(3-methoxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
(1R,2R,4R)-N-{[5-chloro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
N-(6-phenoxypyridin-3-yl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-4-carboxamide
N-cyclopropyl-N-(thiophen-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-(6-chloropyridin-3-yl)-1-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}urea
N-[(3R,4S)-1-[2-hydroxy-6-(trifluoromethyl)pyridine-3-carbonyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
3-(diphenylmethyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,2-oxazole-5-carboxamide
N-[2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(thiophen-2-yl)acetamide
5-benzyl-5-{3-[4-(2-methoxyphenoxy)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
5-propyl-N-(2,2,2-trifluoroethyl)pyrazolo[1,5-a]pyrimidin-7-amine
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl]methanol
N,4-dimethyl-N-[1-(pyridin-4-yl)ethyl]naphthalene-1-carboxamide
methyl (2S)-2-{2-[(3,5-dimethylphenyl)carbamoyl]acetamido}-4-methylpentanoate
1-methyl-2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}azepane
2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-methyl-N-(2-phenylethyl)acetamide
3-[(1-{4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]phenyl}piperidin-4-yl)amino]oxolan-2-one
N-[(6-chloropyridin-3-yl)methyl]-N,4,6-trimethylpyrimidin-2-amine
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)naphthalene-1-carboxamide
2-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}-1,3-thiazole-4-carboxamide
8-[(3-hydroxyphenyl)methyl]-3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(3R,4R)-1-(5-methyl-1,3-thiazole-4-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
(4aS,8aR)-6-[2-(benzyloxy)acetyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
3-{1-[2-(3-chlorophenoxy)propanoyl]piperidin-4-yl}-N-cyclopropylpropanamide
5-(1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}pyrrolidin-2-yl)-3-methyl-1H-1,2,4-triazole
2-[3-oxo-3-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)propyl]-2,3-dihydro-1H-isoindol-1-one
2-[(1-acetylpiperidin-4-yl)oxy]-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-methoxybenzamide
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-(pyrrolidin-3-yl)piperazine
N-{[7-(2-ethylbutanoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-fluorobenzamide
2-[3-(1H-imidazol-1-yl)propyl]-9-[2-(morpholin-3-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one