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2-(2-methoxyethyl)-9-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
7-(4-chlorophenyl)-2-(3-methyl-1H-pyrazol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-(2-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-2-yl}ethyl)phenol
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]pent-4-ynamide
N-(1,2,3-thiadiazol-5-yl)-5-{1-[2-(1H-1,2,4-triazol-1-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-fluoro-N-(2-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]formamido}ethyl)benzamide
4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-{[5-(1H-imidazol-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(6-methylpyrimidin-4-yl)piperidine-4-carboxamide
[(4-{[1-(5-chloro-3-methyl-1H-indole-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl](methyl)(1,2-oxazol-3-ylmethyl)amine
N-[2-(2,4-dichlorophenyl)ethyl]-2-(morpholin-3-yl)acetamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,5-dimethylfuran-3-carboxamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-methyl-N-[3-(morpholin-4-yl)propyl]azepan-4-amine
1-ethyl-N-methyl-N-[(4-phenoxyphenyl)methyl]-1H-pyrazole-5-carboxamide
methyl (2S,4S)-1-(1-benzylpiperidin-4-yl)-4-{2-[4-(trifluoromethyl)phenyl]benzamido}pyrrolidine-2-carboxylate
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-(4-chlorophenyl)-4-[(6-chloropyridin-2-yl)methyl]morpholine
N-[5-({[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)pyrimidin-2-yl]benzenesulfonamide
4,6-dimethyl-3-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
[(3-{[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
1-[(2-methylphenyl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
1-{3-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-phenylprop-2-ynamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N-cyclopentyl-N'-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]butanediamide
{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
2-(2H-1,3-benzodioxol-5-yl)-1-[4-(3-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]ethan-1-one
4-(6-oxopiperidine-3-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
N-(cyclohexylmethyl)-1-cyclopropyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(1-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}-2-[3-(trifluoromethyl)phenyl]ethyl)-N-methylcyclopropanecarboxamide
3-{[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
N-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methylbenzamide
3-[4-(2,4-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
N2-benzyl-N2,7,7-trimethyl-N5-(pyrazin-2-yl)-5,6,7,8-tetrahydroquinazoline-2,5-diamine
1-(1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}piperidin-4-yl)-2-phenylethan-1-ol
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-cyclohexyl-4-[5-(methoxymethyl)furan-2-carbonyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
1-(carbamoylmethyl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidine-3-carboxamide
1-methyl-4-({5-[2-(trimethyl-1H-pyrazol-4-yl)ethyl]-1,2,4-oxadiazol-3-yl}methyl)piperazine
N-{[1-(2,2-dimethylpropyl)piperidin-4-yl]methyl}-2-(pyridin-4-yl)acetamide
2-(4-{[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}phenyl)ethan-1-amine
methyl 5-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-(propane-2-sulfonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
(3S,4S)-3-hydroxy-4-[methyl(quinolin-4-ylmethyl)amino]-N-(2-methylphenyl)pyrrolidine-1-carboxamide
1-[2-methoxy-5-({[2-(2-methylphenyl)ethyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
2-methyl-N-[2-(2-methylpiperidin-1-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
methyl 1-(2-methoxyethoxy)-2-oxo-8-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
2-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}acetamide
N-{[7-(2,3-dimethyl-1H-indole-5-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
1-(1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)-3-methylbutan-1-one