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3-(dimethyl-1H-1,2,4-triazol-1-yl)-N-ethyl-2-methyl-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}propanamide
benzyl({[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl})methylamine
3-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-6-methyl-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridin-4-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
7-(2-methoxyacetamido)-N-(1-methoxypropan-2-yl)-1-methyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
2-[2-(2H-1,3-benzodioxol-5-yl)phenyl]ethan-1-amine
3-[(1-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}pyrrolidin-3-yl)methyl]benzoic acid
2-[9-(furan-3-carbonyl)-7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-ol
5-[(2-ethylpiperidin-1-yl)methyl]-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-ethyl-8-[2-(ethylamino)pyrimidine-5-carbonyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}acetamide
2-(3-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl)propanoic acid
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[(3-methylquinoxalin-2-yl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-[4-(methylsulfanyl)phenyl]-N-{[8-(pyridin-2-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
(4aS,7aR)-1-cyclopentanecarbonyl-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(but-2-yn-1-yl)-N-(furan-2-ylmethyl)-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
1-[2-(4-methoxyphenyl)ethyl]-8-(3-methylbut-2-en-1-yl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}({[4-(trifluoromethoxy)phenyl]methyl})amine
3-methyl-1-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydroquinoxalin-2-one
4-[2-(2-fluorophenyl)acetyl]-1-(4-methylphenyl)piperazin-2-one
N-[(2R,3R)-2-hydroxy-1'-[(2-hydroxy-6-methoxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
N-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyloxan-4-amine
N-methyl-5-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
9-[(6-fluoroquinolin-2-yl)methyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-5-{[(pyridin-3-ylmethyl)amino]methyl}-1H-pyrazole-4-carboxylate
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
N-cyclopropyl-3,4-dimethoxy-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}benzamide
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
N-benzyl-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)acetamide
4-methoxy-3-[1-phenyl-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]benzene-1-sulfonamide
1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
4-hydroxy-4-(5-methylpyridin-2-yl)-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)piperidine-1-carboxamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[3-(4-{[(2,3-difluorophenyl)methyl]amino}piperidin-1-yl)phenyl]-2-methoxybenzamide
5-fluoro-N-methyl-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
2-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-4-(propan-2-yl)-1,3-thiazole
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-2-methoxyacetamide
N-{4-[5-methyl-4-({[3-(trifluoromethyl)phenyl]formamido}methyl)-1,3-oxazol-2-yl]phenyl}pyridine-3-carboxamide
3-[(2-chlorophenyl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-1,2-oxazole-5-carboxamide
2-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1H-1,3-benzodiazole
1-[2-(4-fluorophenyl)piperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-4-(2-phenoxyethyl)piperazine
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[1-(2-methoxyphenyl)ethyl]methylamine
N-[3-(furan-2-yl)propyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
(2S,4R)-4-amino-N-ethyl-1-[(5-ethylpyridin-2-yl)methyl]pyrrolidine-2-carboxamide
1-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)urea
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]acetamide
5-[2-(ethylamino)ethyl]-1-[(3-fluorophenyl)methyl]pyrrolidin-2-one
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-(2-methoxyethyl)-1,4-diazepan-5-one