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4-{[(2,3-dimethoxyphenyl)methyl](ethyl)carbamoyl}benzoic acid
7-(1,3-benzothiazol-2-yl)-4-(2-phenylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(2-methylphenyl)propan-1-one
1-[(5-fluoro-2-methylphenyl)methyl]-5-(2-{[(3-methylphenyl)methyl]amino}ethyl)pyrrolidin-2-one
5-[(2R)-2-hydroxy-2-phenylacetyl]-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-[4-(3-fluorophenyl)phenyl]piperidin-4-amine
1-[3-({[(3-chlorophenyl)methyl]amino}methyl)-7-methylquinolin-2-yl]piperidin-4-ol
N-[(2R,3R)-2-ethoxy-1'-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
3-(4-fluorophenyl)-6-[4-(1H-pyrazol-5-yl)phenyl]pyridazine
3-{2-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]-2-oxoethyl}-1,2,3-oxadiazol-3-ium-5-olate
3-({[3-(morpholin-4-yl)propyl]amino}methyl)-1-(prop-2-en-1-yl)-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
(3R,4S)-4-{[(3,4-dichlorophenyl)methyl](ethyl)amino}oxolan-3-ol
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-2-(1H-pyrazol-1-yl)benzamide
2-{5-[4-(methoxymethyl)-5-methyl-1,2-oxazol-3-yl]-3-(2-phenylethyl)-1H-1,2,4-triazol-1-yl}pyridine
3-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
(1-methyl-1H-imidazol-2-yl)({1-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperidin-4-yl})methanol
4-{5-[1-(1-cyclopropanecarbonylpiperidin-3-yl)-1H-1,2,3-triazol-4-yl]thiophen-2-yl}-2-methylbut-3-yn-2-ol
N-(5-methyl-1,3,4-thiadiazol-2-yl)-4-(pyridin-4-yl)-1,4-diazepane-1-carboxamide
4-methyl-2-(pyrrolidin-1-yl)-6-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyrimidine
(1S,5R)-6-methyl-3-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-4-phenylazepane
6-[9-(cyclopropylmethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl]pyridine-2-carbonitrile
N-(1-cycloheptylpiperidin-3-yl)-3-phenylpropanamide
1-(4-chloro-2-methoxy-5-methylphenyl)-3-methyl-3-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]urea
N-cyclopropyl-1-[(1s,4s)-4-[2-(2-chlorophenoxy)acetamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-(3-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{2-[4-(2-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
(2S)-2-{imidazo[2,1-b][1,3]thiazol-6-ylformamido}-3-(1H-indol-3-yl)propanoic acid
2-[1-(3-fluoropropyl)-1,2,5,6-tetrahydropyridin-3-yl]-N-(furan-2-ylmethyl)piperidine-1-carboxamide
(3aR,6aR)-2-methanesulfonyl-5-[(6-methylquinolin-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{4-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]piperazin-1-yl}pyrazine-2-carbonitrile
1-(2-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(1-benzofuran-2-ylmethyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-acetamido-1-ethyl-N-(2-methoxyethyl)-2-(3-methoxyphenyl)-N-methyl-1H-1,3-benzodiazole-7-carboxamide
1-[2-(3-chlorophenyl)ethyl]-5-{2-[(pyridin-3-ylmethyl)amino]ethyl}pyrrolidin-2-one
methyl 3-{[5-(4-cyclohexylphenyl)-1,2,4-triazin-3-yl]amino}propanoate
1-(4-{[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}phenyl)imidazolidin-2-one
methyl 5-[(3-hydroxy-3-methylbutan-2-yl)amino]-1-methyl-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{[2-(2-aminoethyl)morpholin-4-yl]methyl}-8-fluoroquinolin-4-ol
(2E)-3-(3,4-difluorophenyl)-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}prop-2-enamide
(1-{[methyl({[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl})amino]methyl}cyclopentyl)methanol
N4,6-dimethyl-N4-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyrimidine-2,4-diamine
4-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-1λ6-thiomorpholine-1,1-dione
5-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
[1-(5-chloropyridin-2-yl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
7-(4-methoxy-3-methylbenzoyl)-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3S,4R)-1-(2-aminoethyl)-4-(2,3-dimethoxyphenyl)pyrrolidine-3-carboxylic acid