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N-(2-{[5-acetamido-1-ethyl-2-(3-methoxyphenyl)-1H-1,3-benzodiazol-7-yl]formamido}ethyl)acetamide
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-2,3-dimethoxybenzamide
1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]-N-[2-(methylsulfanyl)ethyl]piperidine-4-carboxamide
3-(3-methylphenoxymethyl)-1-(1H-pyrrole-3-carbonyl)piperidine
5,7-dimethoxy-4-{3-methylimidazo[1,5-a]pyridin-1-yl}-1,2,3,4-tetrahydroquinolin-2-one
2-(3-fluoro-4-methoxyphenyl)-5-(1H-imidazol-1-ylmethyl)pyridine
methyl 4-[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)carbamoyl]butanoate
2-chloro-N-[2-(1,3-thiazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
3-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
5-{[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]amino}-1-(cyclopropylmethyl)azepan-2-one
N-(3-{[(3-hydroxypropyl)[(2-methoxyphenyl)methyl]carbamoyl]amino}phenyl)acetamide
2-methoxy-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetamide
methyl({[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl})[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
2-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyrimidin-4-amine
1-[(1S,5R)-6-(3,5,7-trimethyl-1H-indole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
4-(4-{[3-(1H-1,2,3-benzotriazol-1-yl)propyl]amino}piperidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
8-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{3,5-dimethyl-4-[4-(propan-2-yl)-1,2,3-thiadiazole-5-amido]-1H-pyrazol-1-yl}acetic acid
5-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(thiophen-2-ylmethyl)-1,2,4-oxadiazole
5-(2-chloro-4-methoxyphenoxymethyl)-N-(2-hydroxybutyl)-1H-pyrazole-3-carboxamide
1-methyl-N-{[1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]methyl}-1H-indazole-3-carboxamide
7-chloro-3,5-dimethyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-1-benzofuran-2-carboxamide
1-[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]-2,2-dimethylbutan-1-one
2-methoxy-N-{1-[1-(4-methyl-2-oxopentanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
2-{1-[(5-ethylfuran-2-yl)methyl]piperidine-3-carbonyl}pyridine
2-(8-{[3-(2-hydroxyethoxy)phenyl]methyl}-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl)acetamide
N,N-dimethyl-5-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]pyrrolidin-2-yl}thiophene-2-carboxamide
3-{[(2,2-dimethylpropyl)carbamoyl]methyl}-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-ethyl-3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)pyrrolidine-2,5-dione
1-{2-[2-(4-chlorophenyl)morpholin-4-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
3-[1-(3-chlorothiophene-2-carbonyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
4-(4-methyl-1H-pyrazol-1-yl)-1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperidine-4-carboxylic acid
N-{[7-(3-chlorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-sulfonamide
2-(2-butoxy-4-fluorophenyl)-4-(piperidine-1-carbonyl)pyridine
4-({[(2-methoxyphenyl)methyl](propyl)amino}methyl)benzonitrile
4-[(3aS,6aS)-1-[(6-methylpyridin-2-yl)methyl]-octahydropyrrolo[2,3-c]pyrrol-5-yl]-2-methoxypyridine-3-carbonitrile
ethyl 1-methyl-5-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(ethylamino)-N-[(5-methylpyrazin-2-yl)methyl]pyrimidine-5-carboxamide
1-[1-(4-amino-5-methylpyrimidin-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-({7-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(1H-imidazol-1-yl)acetamide
1-(6-hydroxy-1,4-oxazepan-4-yl)-2-(4-phenylphenyl)ethan-1-one
(3R,9aR)-3-benzyl-8-{[3-(methylsulfanyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N2-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N4,6-dimethylpyrimidine-2,4-diamine
ethyl 1-(2,6-difluorobenzoyl)-3-[(2,4-difluorophenyl)methyl]piperidine-3-carboxylate
4-cyclohexyl-3-{[2-(2,4,5-trimethylphenyl)-1H-imidazol-1-yl]methyl}-4H-1,2,4-triazole
8-(thian-4-yl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
6-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-N-ethyl-N-methylpyridine-3-carboxamide
2-[methyl({5-[5-(trifluoromethyl)pyridin-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)amino]ethan-1-ol