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[(2-fluoro-5-methoxyphenyl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
6-methyl-N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(9H-purin-6-yl)pyrrolidin-3-yl]methanol
3,5-dimethyl-2-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine-1-carbonyl}-1H-indole
methyl 4-[(2-{[4-(4-hydroxyphenyl)piperazin-1-yl]methyl}quinazolin-4-yl)amino]butanoate
2-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-phenylethyl)piperidin-1-yl]methyl}-3-methoxyphenol
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-2-(pyridin-3-ylmethyl)pyrrolidine-1-carboxamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(thiophene-2-sulfonyl)piperidin-3-yl]propanoic acid
2-[(3-methoxyphenyl)methyl]-4-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]morpholine
1-{4-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
(4aR,8aS)-1-[(3,4-dimethoxyphenyl)methyl]-6-[(5-methylthiophen-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
N-({8-[(2-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-3-methylbutanamide
1-(4-chlorophenyl)-5-methyl-4-[3-(1H-pyrrol-1-yl)propanoyl]piperazin-2-one
1-(2-aminoethyl)-N-cyclohexyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-(2-{[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}ethyl)azepane
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[3-(1H-indazol-1-yl)propyl]acetamide
1-(2-amino-9H-purin-6-yl)-4-phenoxypiperidine-4-carboxylic acid
N-methyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyridin-2-amine
1-(2-methoxy-4-{[(3-methylbutyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methylacetamide
3-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidine-1-carbonyl}pyridin-1-ium-1-olate
{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(isoquinolin-5-ylmethyl)methylamine
[(4-{1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-2-yl}phenyl)methyl]dimethylamine
methyl 3-acetamido-1-(3-methylbutyl)-5-{[(2,4,6-trimethoxyphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]furan-2-carboxamide
1-ethyl-4-(4-{4-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]piperidin-1-yl}benzoyl)piperazine
N-(2,3-dihydro-1H-inden-1-yl)-2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
4-{2-oxo-4-[3-(pyridin-4-yl)propanoyl]piperazin-1-yl}benzonitrile
N,N-dimethyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]aniline
(3aR,6aR)-2-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methyl-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-4-(4-methylphenyl)piperazine
7-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(2-fluorophenyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,2,4-triazin-3-amine
1-[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
1-(oxan-4-ylmethyl)-4-[(1R,2R)-2-phenylcyclopropanecarbonyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
3-(4-methoxyphenyl)-N-methyl-N-(thiophen-3-ylmethyl)propanamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-(1-propylcyclopropyl)acetamide
N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]thiophene-3-carboxamide
1-(cyclohexylmethyl)-3-hydroxy-3-{[(2-methylpropyl)amino]methyl}piperidin-2-one
N-(1-{1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperidin-4-yl}-2-(2,4-difluorophenyl)ethyl)-N-methylpropanamide
N-[1-(4-{[(1-phenylcyclopentyl)methyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]oxane-4-carboxamide
2-{4-[3-(benzyloxy)piperidine-1-carbonyl]piperidin-1-yl}-4-methylquinazoline
1-[(4aR,8aR)-7-[(4-chloro-3-fluorophenyl)methyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
N-{[7-(1H-indole-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
N-methyl-5-(propan-2-yl)-N-(quinolin-5-ylmethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3,3-diethyl-1-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}pyrrolidine
4-[(4-fluoro-3-methoxyphenyl)methyl]-1-(2-methylphenyl)piperazin-2-one