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{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)[(3-methyl-1H-pyrazol-5-yl)methyl]amine
4-{[6-(methoxymethyl)pyrimidin-4-yl]amino}-1-propylpyrrolidin-2-one
4-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
1-[1-(3-methoxypropanoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N,N-dimethyl-2-[methyl({[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl})amino]propanamide
(2S,4R)-4-amino-1-(4-amino-6-fluoroquinoline-3-carbonyl)-N-methylpyrrolidine-2-carboxamide
4-benzyl-3-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(3-chlorophenyl)-N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-3-phenylpropanamide
(2R)-1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxy-2-phenylethan-1-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-2-(furan-2-yl)-N-methyl-2-oxoacetamide
5-fluoro-N-(2-methoxyethyl)-1,3-dimethyl-N-[(5-methylthiophen-2-yl)methyl]-1H-indole-2-carboxamide
methyl 6-(4-chlorobenzoyl)-2-[(prop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(1-methyl-1H-imidazol-2-yl)piperidine
1-[(5-phenylthiophen-2-yl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-methyl-N-[2-(5-methylfuran-2-yl)ethyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
[1-(2H-1,3-benzodioxol-4-ylmethyl)-3-[(2-fluorophenyl)methyl]piperidin-3-yl]methanol
3-(2,3-dihydro-1H-inden-2-yl)-8-[(2-hydroxy-5-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-(2-amino-6-methoxypyrimidin-4-yl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-N-ethylacetamide
{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(1-methoxypropan-2-yl)amine
2-[1-benzyl-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N,N-diethylacetamide
[(8-chloroquinolin-2-yl)methyl][(3-ethyl-1,2-oxazol-5-yl)methyl]methylamine
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}cyclopropanamine
8-cyclobutyl-3-ethyl-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
3-{1-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}-1,2-dihydroquinolin-2-one
4-chloro-3-{[(5-oxo-1-propylpyrrolidin-3-yl)carbamoyl]amino}-N-(propan-2-yl)benzamide
1-[(2-fluorophenyl)methyl]-N-[(3-methylpyridin-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-{4-[(4-methyl-1,4-diazepan-1-yl)methyl]phenyl}-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-(dimethylamino)butan-1-one
2-(2-methoxyethyl)-8-(4-methylpent-3-en-1-yl)-2,8-diazaspiro[5.5]undecan-3-one
{3-[(1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]phenyl}methanol
2-[4-phenyl-5-(2-phenylethyl)-1H-imidazol-1-yl]-1-(pyridin-3-yl)ethan-1-ol
1-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-{[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
6-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-N-{[3-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
N-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-(pyridin-3-ylmethyl)piperidin-4-amine
2-(hydroxymethyl)-N-[4-(2-methoxyphenyl)phenyl]piperidine-1-carboxamide
2-{8-[(3-ethoxy-4-methoxyphenyl)methyl]-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
4-(5-methylpyridin-2-yl)-1-[3-(1H-pyrazol-4-yl)benzoyl]piperidin-4-ol
N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-[4-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)piperazin-1-yl]-1,3-benzoxazole
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[3-(morpholin-4-yl)propyl]acetamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-4-amine
5-cyclobutyl-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1,3,4-oxadiazol-2-amine
N-benzyl-3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(2-hydroxyethyl)propanamide
1-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
1,3-dimethyl-2,6-dioxo-N-[1-(thian-4-yl)piperidin-4-yl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[(1r,4r)-4-hydroxycyclohexyl]acetamide
1-benzyl-5-{[(4-fluorophenyl)methyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide