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1-methyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-({7-[2-(cyclohex-1-en-1-yl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(pyrimidin-2-ylsulfanyl)acetamide
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide
3-(2-oxo-2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}ethyl)-4-(2-phenylethyl)piperazin-2-one
(2R)-2-cyclohexyl-2-hydroxy-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
4-(pyridin-2-yl)-N-[3-(pyridin-2-yl)propyl]pyrimidin-2-amine
6-ethoxy-2-{4-[2-(4-fluorophenyl)piperidine-1-carbonyl]piperidin-1-yl}-4-methylquinazoline
5-ethyl-2,4-dimethyl-6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
(1-{3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidin-4-yl)(thiophen-2-yl)methanol
9-methoxy-3-(naphthalen-2-ylmethyl)-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[5-(2,4,6-trimethylphenyl)pyridin-2-yl]methanesulfonamide
1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-ethylpiperazine
7-chloro-3-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinolin-4-ol
N-{[5-chloro-7-(1H-indol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylpropanamide
1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-4-(piperidine-1-carbonyl)piperidine
1-[(2-fluorophenyl)methyl]-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-sulfamoylbenzamide
3-[(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amino]-N-(thiophen-2-ylmethyl)propanamide
6-(3-methoxypyrazin-2-yl)-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
methyl 4-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-oxo-6-(pyridin-4-ylmethoxy)-1,4-diazepane-1-carbonyl}benzoate
{3-ethyl-1-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidin-3-yl}methanol
5-butyl-1'-(2-methylpyrimidine-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
4-(1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-3,5-dimethyl-1,2-oxazole
4-{[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
7-[2-(2-methoxyphenyl)acetyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-{4-[3-(2-phenylethyl)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
5-{[2-(dimethylamino)-2-(2-methylphenyl)acetamido]methyl}-1,2,4-oxadiazole-3-carboxamide
(2S)-2-{[2-(3-ethoxyphenoxy)ethyl]amino}-3-methylbutanamide
4-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
4-(4-chloro-1-ethyl-1H-pyrazole-5-carbonyl)-2-(4-chlorophenyl)morpholine
1-[1-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
5-(5-methyl-1-phenyl-1H-pyrazol-4-yl)-4-phenyl-1-(pyrrolidin-3-yl)-1H-imidazole
N-[(3,4-dimethoxyphenyl)methyl]-4-methoxy-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
7-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
4-[5-(piperidine-1-carbonyl)-1H-pyrrol-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
(3S,9aR)-8-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-(5-chloro-2-methylbenzoyl)-3-(3-methoxypropyl)piperidine
3-chloro-4-{[1-(cyclopentylmethyl)piperidin-4-yl]oxy}-N-[2-(dimethylamino)ethyl]benzamide
2-(2,6-difluorophenyl)-1-{1-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-azaspiro[2.5]octan-6-yl}ethan-1-one
2-{3-cyclopentyl-5-[2-(ethylamino)-4-methyl-1,3-thiazol-5-yl]-1H-1,2,4-triazol-1-yl}acetic acid
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]{[5-(oxan-2-yl)furan-2-yl]methyl}amine
1-{[3-(2-butylpyrrolidine-1-carbonyl)-1H-pyrazol-5-yl]methyl}-1H-1,3-benzodiazole
N,N-dimethyl-2-{2-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}ethane-1-sulfonamide
N-[(1-hydroxycyclohexyl)methyl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
ethyl 5-(2,3-dihydro-1H-inden-2-yl)-1-[2-(dimethylamino)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-7-methylimidazo[1,2-a]pyridine-2-carboxamide