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2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]acetamide
(4aS,7aR)-1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[4-(3,5-dimethyl-1-benzofuran-2-carbonyl)piperazin-1-yl]ethan-1-ol
methyl 1-[(3R,5S)-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(3aS,6aS)-2-cyclopentyl-5-(2,6-dimethylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl 3-[(3-methoxyphenyl)methyl]-1-(2-methoxypyridine-3-carbonyl)piperidine-3-carboxylate
2-methoxy-N-[(2R,3R)-1'-[(4-methoxy-3-methylphenyl)methyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}({[3-(methylsulfanyl)phenyl]methyl})(pyridin-4-ylmethyl)amine
3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1H-indazole
2-ethyl-4-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-6-methylpyrimidine
(4-methyl-5-{[1-(4,4,4-trifluorobutyl)piperidin-4-yl]methyl}-4H-1,2,4-triazol-3-yl)methanol
(5S,9aS,9bS)-5-[4-(1H-pyrazol-1-yl)phenyl]-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[(3R,4S)-1-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
2-(4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-(2-methylpropyl)piperazin-2-yl)ethan-1-ol
dimethyl[(4-{[5-(piperidine-1-carbonyl)pyridin-2-yl]oxy}phenyl)methyl]amine
N-[2-(3-methoxyphenyl)-1-{1-[2-(2-methoxyphenyl)acetyl]piperidin-4-yl}ethyl]-N-methylcyclopropanecarboxamide
3-{5-[(2-aminopyridin-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(morpholin-4-yl)propan-1-one
N-({5-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]pyridine-4-carboxamide
1-(1-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)-2-(3-methoxyphenyl)ethan-1-one
4-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]phenol
4-{[3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)carbamoyl}-3,5-dimethyl-1H-pyrrole-2-carboxylic acid
2,3,6-trifluoro-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
6-[4-(2,5-dihydro-1H-pyrrol-1-yl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-N4-methylpyrimidine-2,4-diamine
1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
N-[3-(4-{[3-(4-methoxyphenyl)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-5-methylthiophene-2-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[(thian-4-yl)amino]pyrrolidin-2-one
1-(2,1,3-benzoxadiazol-4-ylmethyl)-N-(4-fluorophenyl)piperidin-3-amine
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-3-methylthiophene-2-carboxamide
(3S,4R)-1-[(5-ethylpyridin-2-yl)methyl]-4-methyl-3-(2-methylpropyl)piperidin-4-ol
5-[(diethylamino)methyl]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methylfuran-3-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-3,3,3-trifluoro-N-methylpropanamide
N,N-diethyl-3-(1-hydroxy-3-methylbutan-2-yl)-5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
3-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1-(1-propyl-1H-pyrazol-5-yl)urea
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
1-(4-ethylpiperazin-1-yl)-3-(3-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
1-{4-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
3-[(3R,4S)-1-(3,4-dimethylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
3-[(3-methoxyphenyl)methyl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
N-[2-(4-fluorophenyl)-1-[1-(quinolin-8-ylmethyl)piperidin-4-yl]ethyl]-N-methyl-3-(methylsulfanyl)propanamide
1-(2-methoxyphenyl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
N-ethyl-2-{[2-(ethylamino)pyrimidin-5-yl]formamido}propanamide
2-({1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-4-yl}oxy)pyrimidine
1-[(3-fluorophenyl)methyl]-4-[(6-methoxy-1H-indazol-3-yl)methyl]piperazin-2-one
1'-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)-3,5-dimethyl-1,2-oxazole-4-sulfonamide