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N-[3-(furan-2-yl)propyl]-1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-amine
7-(3-methyl-1H-pyrazole-5-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
8-[3-(ethylsulfanyl)propanoyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-ethyl-2-methyl-N-[3-(morpholin-4-yl)propyl]pyrimidin-4-amine
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]-2-(1,1,2,2-tetrafluoroethoxy)benzamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
4-cyclobutaneamido-N-methyl-N-[2-(pyrrolidin-1-ylmethyl)propyl]benzamide
3-{1-[(2,6-difluoro-3-methoxyphenyl)methyl]-1H-imidazol-2-yl}phenol
1-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-2-ethylpiperidine
4-[(3-chlorophenyl)methyl]-1-(2,3-difluorobenzoyl)-1,4-diazepan-5-one
3-hydroxy-3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-1-(3-phenylpropyl)piperidin-2-one
2-(2-{3,9-diazaspiro[5.6]dodecan-9-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-(2-methoxyethyl)-1-[1-(3-methylpyrazin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
ethyl 4-[(4-{[1-(pyridine-4-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
5-[4-(2-chlorophenyl)piperazine-1-carbonyl]-1-methyl-1H-pyrrole-3-carbonitrile
5-methoxy-2-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]-1,4-dihydropyridin-4-one
2-{4-[(8-fluoroquinolin-2-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
3-hydroxy-1-(2-methoxyethyl)-3-({[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)piperidin-2-one
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-oxo-2,3-dihydro-1H-indene-1-carboxamide
N-methyl-N-{[1-(2-methylphenyl)-1H-1,2,3,4-tetrazol-5-yl](phenyl)methyl}-1,2-oxazole-3-carboxamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-(methylsulfanyl)-N-(oxolan-2-ylmethyl)propanamide
3-(2-chlorophenyl)-N-{[5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
2-[2-(3-phenylpiperidin-1-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
6-[3-(1H-pyrazol-5-yl)phenyl]pyridine-3-carbonitrile
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyrimidin-2-ylsulfanyl)acetamide
N-[(3-methyl-7-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(thiophen-3-yl)acetamide
2-(4-chlorophenyl)-4-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}morpholine
4-methoxy-N-(2-methoxyethyl)-2-({1-[(2,4,5-trimethylphenyl)methyl]piperidin-4-yl}oxy)benzamide
N-[(3,4-dimethoxyphenyl)methyl]-2-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]acetamide
3-{1-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]piperidin-4-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl[1-(pyridin-2-yl)ethyl](4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
3-chloro-N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropylbenzamide
1-(diethylamino)-3-(2-methoxy-4-{[(2-methylpropyl)amino]methyl}phenoxy)propan-2-ol
2-[(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenol
3-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazine
2-[(2,6-dichlorophenyl)methyl]-6-(piperidin-3-yl)-3,4-dihydropyrimidin-4-one
4-({2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl}methyl)-1-methyl-1H-pyrrole-2-carbonitrile
2,3-dimethyl-6-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
3-{2-[3-(2-chlorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-(3-methoxypropyl)pyrrolidine-2,5-dione
N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-(pyrazin-2-yl)propanamide
3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]propanamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-(1H-1,3-benzodiazole-5-carbonyl)-1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-cyclopropyl-6-[4-(pyridin-2-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,3-benzoxazole
(2S,4R)-1-{[4-(benzyloxy)phenyl]methyl}-4-[(4-fluorophenyl)sulfanyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
6-methyl-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}imidazo[2,1-b][1,3]thiazole-5-carboxamide
5-ethyl-N-{[8-(4-fluorobenzoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1,2-oxazole-3-carboxamide
1-[(2,6-difluorophenyl)methyl]-4-[2-(4-methyl-1,4-diazepane-1-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol