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N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-4-(piperidin-1-yl)butanamide
(3S,4S)-4-cyclopropyl-1-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}pyrrolidine-3-carboxylic acid
4-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]-4-oxobutane-1-sulfonamide
5-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazole
3-fluoro-2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine
2-methyl-5-(4-{[(3-phenylcyclobutyl)amino]methyl}piperidin-1-yl)-2,3-dihydropyridazin-3-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5-methoxyfuran-2-carboxamide
1-(3-methoxyphenyl)-3-methyl-4-[3-(pyridin-3-yl)propanoyl]piperazin-2-one
1-[(3aS,6aS)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-octahydropyrrolo[2,3-c]pyrrol-5-yl]-2-(furan-2-yl)ethane-1,2-dione
5-({ethyl[(4-ethylphenyl)methyl]amino}methyl)-N-(propan-2-yl)pyrimidin-2-amine
N-[(2R,3R)-1'-[(3,5-dimethoxyphenyl)methyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
2-{1-[(2-fluorophenyl)methyl]-4-(isoquinolin-5-ylmethyl)piperazin-2-yl}ethan-1-ol
ethyl 4-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]butanoate
N-(naphthalen-1-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(cyclopropylmethyl)-5-[(4-fluorophenyl)methyl]-5-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
2-{1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}propan-2-ol
N-{1-[1-(3,4-difluorobenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylpyridine-3-carboxamide
4-{1-[(4-methoxyphenyl)methyl]piperidin-3-yl}-5-phenyl-2-(pyridin-4-yl)pyrimidine
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3-methyl-1-phenyl-1H-pyrazole
6-(2H-1,3-benzodioxole-5-carbonyl)-1-(cyclopropylmethyl)-3-(2-methylquinolin-5-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(3S,9aR)-8-(4-chlorobenzenesulfonyl)-3-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[1-(dimethylamino)-2-methylpropan-2-yl]-6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}({2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl})amine
7-(2-methoxyethyl)-2-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
N-[5-(2-ethoxyethyl)-1,3,4-thiadiazol-2-yl]-3-(4-fluorophenoxy)piperidine-1-carboxamide
4-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-methylpiperazin-2-one
benzyl[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl](1,3-thiazol-2-ylmethyl)amine
4-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-{4-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
(4aR,7aS)-1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclohexyl-4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
N-[4-(propylsulfamoyl)phenyl]-3-(pyridin-2-yl)azetidine-1-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(piperidin-1-yl)acetamide
3-[5-(3-phenyl-1,2,4-oxadiazol-5-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
N-methyl-9-oxo-N-[1-(1,3-thiazol-2-yl)ethyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
5-ethyl-2,6-dimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyrimidin-4-amine
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
6-[2-hydroxy-2-(3-methoxyphenyl)ethyl]-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
3-(1-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-1H-1,2,3-triazol-4-yl)benzonitrile
1-(2-methoxyacetyl)-N-[3-(3-methylphenyl)phenyl]pyrrolidine-2-carboxamide
5-chloro-N-(2-hydroxyethyl)-3-phenyl-N-propyl-1H-indole-2-carboxamide
7-methoxy-4-methyl-2-{4-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]piperidin-1-yl}quinazoline
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
3-methyl-3-(2-oxo-2-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethyl)-2H,3H-imidazo[1,2-a]pyridin-2-one
N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pent-4-enamide
N-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]furan-3-carboxamide
1-{5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
1-(oxan-4-yl)-4-(1H-pyrrole-2-carbonyl)-1,4-diazepan-6-ol
4-hydroxy-2-(4-methylphenyl)-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}pyrimidine-5-carboxamide