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(2-chloro-6-fluorophenyl)({4-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl})methanol
2-{1-[cyclopropyl(6-methylpyridin-2-yl)methyl]-1H-imidazol-2-yl}-1-methyl-1H-1,3-benzodiazole
methyl 3-[2-(4-methylphenoxy)acetyl]-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-(2,2-dimethyloxane-4-carbonyl)-1-(4-methoxyphenyl)piperazin-2-one
(3R,4R)-3-cyclopropyl-4-methyl-1-(1,2-thiazole-5-carbonyl)pyrrolidin-3-ol
1-[4-(morpholin-4-yl)-3-(pyridin-4-yl)phenyl]ethan-1-one
2-[2-(2-fluoro-4-methoxyphenyl)-1H-imidazol-1-yl]-N-(2-methylphenyl)acetamide
(3S,4R)-3-benzyl-1-(2,6-dimethylbenzoyl)-4-methylpiperidin-4-ol
1-(5-chloro-2-methylphenyl)-4-{3-[(4-fluorophenyl)methyl]-1,2-oxazole-5-carbonyl}piperazine
N-(2-{[1-(propan-2-yl)piperidin-4-yl]formamido}ethyl)pyridine-4-carboxamide
1-{4-[(dimethylsulfamoyl)amino]phenyl}-N-[3-(furan-2-yl)-3-phenylpropyl]piperidin-4-amine
4-ethyl-1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
[(3,4-dimethoxyphenyl)methyl](methyl){[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1H-imidazole-2-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(3-fluoropyridin-4-yl)pyrrolidin-3-yl]methanol
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(morpholin-4-yl)ethan-1-one
1-{1-[(4-chlorophenyl)methyl]-3-(ethoxymethyl)-1H-1,2,4-triazol-5-yl}cyclopropane-1-carboxamide
(2R,6S)-4-{1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-4-yl}-2,6-dimethylmorpholine
2-(5-methylfuran-2-yl)-1-[(2-methyloxolan-2-yl)methyl]-1H-imidazole
1-ethyl-3-{2-[2-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(3-methylphenyl)ethan-1-one
5-{[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(3-ethoxypropyl)propanamide
2-methyl-1-(4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)propan-1-ol
3-hexyl-8-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(4-fluoro-2-methoxyphenyl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]acetic acid
5-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}-2-(pyridin-3-yl)pyrimidine
3-chloro-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]benzamide
6-[(3-hydroxyazetidin-1-yl)methyl]-2-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-dihydropyridine-3-carboxamide
1-(2-aminoethyl)-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
1-[(3-methoxyphenyl)methyl]-N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-6-oxopiperidine-3-carboxamide
7-chloro-4-{2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-N-[1-(naphthalen-1-yl)ethyl]acetamide
N-[(2R,3R)-1'-(2-hydroxy-4-methoxybenzoyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
3-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]-N-(pyridin-3-yl)propanamide
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-(pyridin-2-ylmethyl)piperazine
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidine
2-methyl-4-[4-(1-methylpiperidin-4-yl)piperidin-1-yl]pyridine
1-{[4-(2H-1,3-benzodioxol-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
1-{3-[4-({[2-(4,6-dimethylpyrimidin-2-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
N-cyclopropyl-4-(4-fluorophenyl)-N-{[4-methoxy-3-(pyridin-4-ylmethoxy)phenyl]methyl}benzamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-[(4-fluorophenyl)methyl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
2-methoxy-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}pyridine-4-carboxamide
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)cyclopentanecarboxamide
N-[(3S,4R)-4-(4-methylphenyl)-1-(6-methylpyridine-2-carbonyl)pyrrolidin-3-yl]cyclopropanecarboxamide
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-4-(thiophen-2-yl)butanamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidine-3-carboxamide
1-(2,6-difluoro-3-methylbenzoyl)-2-[2-(thiophen-2-yl)ethyl]piperidine
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-[(2-hydroxyethyl)sulfanyl]-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide