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[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
3-{4-[1-(pyrimidin-5-ylmethyl)pyrrolidin-3-yl]pyridin-2-yl}quinoline
1-[(2-chlorophenyl)methyl]-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-1H-1,2,3-triazole-4-carboxamide
1-[(2-fluorophenyl)methyl]-4-[2-methyl-2-(morpholin-4-yl)propyl]-1,4-diazepane
2-(1H-imidazol-1-yl)-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)ethan-1-one
1-[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-(thiophen-2-yl)ethan-1-one
9-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-fluoro-N-({1-[(2E)-2-methylbut-2-en-1-yl]piperidin-3-yl}methyl)benzamide
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{[methyl(oxan-4-yl)amino]methyl}-N-(1-oxo-2,3-dihydro-1H-inden-5-yl)benzamide
benzyl (7R,9aR)-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
2-(2-{1-[3-(3-methoxyphenyl)propanoyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
2-[2-(4-ethylpiperazin-1-yl)-2,3-dihydro-1H-indene-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1-[3-(benzyloxy)piperidin-1-yl]-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propan-1-one
1-(1H-indazol-6-yl)-5-methyl-4-{7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carbonyl}piperazin-2-one
4-chloro-N-(propan-2-yl)-3-({[2-(1H-pyrazol-4-yl)ethyl]carbamoyl}amino)benzamide
6-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoxaline
3-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(pyrimidin-2-yl)piperidine-4-carboxylic acid
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(2-methylphenyl)methyl]-N-propyl-1,2-oxazole-3-carboxamide
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2-propylpyridine-4-carboxamide
6-fluoro-4-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-1,2-dihydroquinolin-2-one
1-{1-[6-(2-fluorophenyl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
N-{[2-methoxy-5-(1H-pyrazol-4-yl)phenyl]methyl}cyclopentanamine
N-({1-[(3,5-dimethoxyphenyl)methyl]piperidin-3-yl}methyl)-2-(4-methoxyphenyl)acetamide
N-methyl-N-(2-methylpropyl)-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-(2-phenylpropyl)benzamide
1-[(2-fluorophenyl)methyl]-N-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-N-methylpiperidin-3-amine
8-[(2S)-2-aminohexanoyl]-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
6-[(4-fluorophenyl)methoxy]-1-(propan-2-yl)-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1,4-diazepan-2-one
N-methyl-3-[(morpholine-4-carbonyl)amino]-N-phenylazepane-1-carboxamide
ethyl 4-{6-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate
1-(diethylamino)-3-{4-[(4,4-difluoropiperidin-1-yl)methyl]-2-methoxyphenoxy}propan-2-ol
3-{2-[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]ethyl}-1,3-oxazinan-2-one
N-(prop-2-en-1-yl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N-[(4-chlorophenyl)(pyridin-4-yl)methyl]oxolane-2-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-1-(3-phenylpropyl)-N-(prop-2-en-1-yl)-1H-1,2,3-triazole-4-carboxamide
N-[(5-fluoro-2-methylphenyl)methyl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-({8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)oxane-4-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[(3S)-2-oxoazepan-3-yl]benzamide
5-[1-(but-2-ynoyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
N-[(2R,3R)-1'-[2-(4-chlorophenoxy)acetyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-[(3,4-difluorophenyl)methyl]-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{1-cyclohexyl-4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
8-[(2-methyl-1H-indol-3-yl)methyl]-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methyl-4-[3-(4H-1,2,4-triazol-4-yl)phenyl]pyrimidine
N,1-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
2-(2-phenylpyrimidin-4-yl)pyridine-4-carboxylic acid
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-phenylethan-1-one